| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3125728 | 18 | Activity | = | 102 | % | ALA3132644 | % | Homo sapiens | |||
| 2. |  ALA3125727 | 19 | Activity | = | 103 | % | ALA3132644 | % | Homo sapiens | |||
| 3. |  ALA3125726 | 20 | Activity | = | 105 | % | ALA3132644 | % | Homo sapiens | |||
| 4. |  BAY-091 | EUB0001564 | % inhibition | 8.28 | % | ALA4888125 | Not Active | % | Homo sapiens | |||
| 5. |  Defactinib | DEFACTINIB | % inhibition | 13 | % | ALA4887113 | Not Active | % | Homo sapiens | |||
| 6. |  ALA2180408 | Figure 27, R1C1 | % inhibition | 0 | % | ALA4886206 | Not Active | % | Homo sapiens | |||
| 7. |  ALA4580220 | EUB0000311 | % residual kinase activity | 110 | % | ALA4884253 | Not Active | % | Homo sapiens | |||
| 8. |  TC-S 7001 | SID103905649 | % inhibition | 9 | % | ALA4881502 | Not Active | % | Homo sapiens | |||
| 9. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 96 | % | ALA4880989 | Not Active | % | Homo sapiens | |||
| 10. |  2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | % inhibition | -25 | % | ALA4880588 | Not Active | % | Homo sapiens | |||
| 11. |  ALA5201686 | 10f | Activity | > | 75 | % | ALA5158110 | % | Homo sapiens | |||
| 12. |  Vorinostat (SAHA, MK0683) | SAHA | IC50 | 0 | ALA4845114 | Not Determined | Homo sapiens | |||||
| 13. |  Tubastatin A | Tubastatin A | IC50 | 0 | ALA4845114 | Not Determined | Homo sapiens | |||||
| 14. |  ALA4877598 | 8b-P | IC50 | > | 1000 | nM | ALA4845114 | nM | Homo sapiens | |||
| 15. |  ALA4859978 | 8b-N | IC50 | = | 68.2 | nM | ALA4845114 | 7.17 | nM | Homo sapiens | ||
| 16. |  ALA4867598 | 8b | IC50 | = | 27.2 | nM | ALA4845114 | 7.57 | nM | Homo sapiens | ||
| 17. | Vorinostat (SAHA, MK0683) | SAHA | INH | = | 0.8 | % | ALA4845098 | % | Homo sapiens | |||
| 18. |  ALA216543 | SID124880405 | INH | = | 46.6 | % | ALA4845098 | % | Homo sapiens | |||
| 19. |  ALA1276127 | Indirubin | INH | = | 25.1 | % | ALA4845098 | % | Homo sapiens | |||
| 20. |  ALA4852087 | 8f | INH | = | -2.7 | % | ALA4845098 | % | Homo sapiens |
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