# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2377825 | 51 | IC50 | = | 6.6 | nM | ALA2380178 | 8.18 | nM | Homo sapiens | ||
2. | Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 2.9 | nM | ALA2380178 | 8.54 | nM | Homo sapiens | ||
3. | ALA2377825 | 51 | INH | = | 80 | % | ALA2380163 | % | Homo sapiens | |||
4. | ALA2333445 | 1 | Activity | = | 96 | % | ALA2349834 | % | Homo sapiens | |||
5. | ALA2312140 | 1 | INH | >= | 80 | % | ALA2316984 | % | Homo sapiens | |||
6. | ALA2312142 | 3 | INH | = | 50 | % | ALA2316984 | % | Homo sapiens | |||
7. | ALA3288908 | 15f | INH | = | -17 | % | ALA3294071 | % | Homo sapiens | |||
8. | ALA3288908 | 15f | INH | = | -1 | % | ALA3294070 | % | Homo sapiens | |||
9. | Staurosporine (DMSO solution) | 1 (Staurosporine) | INH | = | -90 | % | ALA3294069 | % | Homo sapiens | |||
10. | ALA3288908 | 15f | INH | = | 2 | % | ALA3294069 | % | Homo sapiens | |||
11. | BI 605906 | BI605906 | % Ctrl | 100 | % | ALA4887263 | Not Active | % | Homo sapiens | |||
12. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 88 | % | ALA4883858 | Not Active | % | Homo sapiens | |||
13. | ALA213805 | CA224 | INH | 0 | ALA3375312 | Not Active | % | Homo sapiens | ||||
14. | Palbociclib | 43(table 3) | IC50 | = | 0.016 | uM | ALA4480963 | 7.80 | nM | Homo sapiens | ||
15. | Palbociclib | 43(table 3) | IC50 | = | 0.018 | uM | ALA4480908 | 7.75 | nM | Homo sapiens | ||
16. | ALA4542308 | 50 | IC50 | > | 100 | uM | ALA4480908 | nM | Homo sapiens | |||
17. | ALA4578017 | 40; Cink4T | IC50 | > | 100 | uM | ALA4480908 | nM | Homo sapiens | |||
18. | ALA4561548 | 34 | IC50 | > | 100 | uM | ALA4480908 | nM | Homo sapiens | |||
19. | ALA4061054 | 5p | IC50 | > | 100 | uM | ALA4480908 | nM | Homo sapiens | |||
20. | Palbociclib | 43(table 3) | INH | = | -97 | % | ALA4480903 | % | Homo sapiens |