# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI 605906 | BI605906 | % Ctrl | 68.6 | % | ALA4887631 | Not Active | % | Homo sapiens | |||
2. | ALA4574669 | (R,R)-36n | INH | 0 | ALA4351807 | Not Active | % | Homo sapiens | ||||
3. | ALA4465324 | 11 | Activity | = | 64 | % | ALA4339893 | % | Homo sapiens | |||
4. | ALA4465324 | 11 | Activity | = | 22 | % | ALA4339892 | % | Homo sapiens | |||
5. | D4476 | K00219, D4476 | IC50 | = | 0.3 | uM | ALA4336769 | 6.52 | nM | Homo sapiens | ||
6. | N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamide | CK1-7 | IC50 | = | 9.5 | uM | ALA4336766 | 5.02 | nM | Homo sapiens | ||
7. | ALA4588446 | 7, 19 | INH | = | 77 | % | ALA4331914 | % | Homo sapiens | |||
8. | ALA4460272 | 6 | INH | = | 0 | % | ALA4331973 | % | Homo sapiens | |||
9. | ALA4589022 | 32 | INH | = | 0 | % | ALA4331973 | % | Homo sapiens | |||
10. | ALA4524629 | 18 | INH | = | 86 | % | ALA4331914 | % | Homo sapiens | |||
11. | ALA4449552 | 4 | INH | = | 46 | % | ALA4331914 | % | Homo sapiens | |||
12. | ALA4440433 | 9 | INH | = | 27 | % | ALA4331914 | % | Homo sapiens | |||
13. | ALA4557538 | 3c; SKLB0533 | Activity | = | 106.5 | % | ALA4314813 | % | Homo sapiens | |||
14. | ALA5172397 | 36; TUL01101 | Activity | = | 102 | % | ALA5154577 | % | Homo sapiens | |||
15. | ALA5192780 | C20 | INH | < | 25 | % | ALA5107255 | % | Homo sapiens | |||
16. | CX-4945 (Silmitasertib) | 25n | IC50 | = | 4 | nM | ALA5055513 | 8.40 | nM | Homo sapiens | ||
17. | (+)-JQ1 | (+)-JQ1 | IC50 | 0 | ALA5055513 | Not Determined | Homo sapiens | |||||
18. | ALA5091216 | 44e | IC50 | = | 230 | nM | ALA5055513 | 6.64 | nM | Homo sapiens | ||
19. | ALA1782169 | 7a | IC50 | > | 10 | uM | ALA5227428 | nM | Homo sapiens | |||
20. | ALA1782170 | 7b | IC50 | > | 10 | uM | ALA5227428 | nM | Homo sapiens |