# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (E)-Guggulsterone | E-guggulsterone (1b) | IC50 | > | 100 | uM | ALA4374497 | nM | Homo sapiens | |||
2. | (E)-Guggulsterone | E-guggulsterone (1b) | EC50 | > | 100 | uM | ALA4374496 | nM | Homo sapiens | |||
3. | ALA4449687 | 11 | IC50 | = | 32.4 | uM | ALA4332166 | 4.49 | nM | Homo sapiens | ||
4. | Tegatrabetan (BC-2059) | 14, BC-2059 | INH | 0 | ALA3603649 | Not Active | % | Homo sapiens | ||||
5. | Tegatrabetan (BC-2059) | 14, BC-2059 | INH | 0 | ALA3603648 | Not Active | % | Homo sapiens | ||||
6. | ALA2348874 | 3{1,18} | INH | 0 | ALA2352072 | Dose-dependent effect | % | Homo sapiens | ||||
7. | ALA2349059 | NH3, NH-3 | INH | 0 | ALA2352072 | Active | % | Homo sapiens | ||||
8. | ALA3763166 | 40 | INH | < | 50 | % | ALA3766993 | % | Homo sapiens | |||
9. | ALA594025 | 5, PF-00277343 | EC50 | = | 0.5 | nM | ALA1068517 | 9.30 | nM | Homo sapiens | ||
10. | ALA252358 | 2d | Activity | = | 1 | % | ALA926597 | % | Homo sapiens | |||
11. | ALA255069 | 2f | Activity | = | 0 | % | ALA926597 | % | Homo sapiens | |||
12. | ALA399093 | 3c | Activity | = | 0 | % | ALA926597 | % | Homo sapiens | |||
13. | ALA254234 | 3d | Activity | = | 4 | % | ALA926597 | % | Homo sapiens | |||
14. | ALA254235 | 3e | Activity | = | 0 | % | ALA926597 | % | Homo sapiens | |||
15. | ALA398653 | 3f | Activity | = | 0 | % | ALA926597 | % | Homo sapiens | |||
16. | ALA398654 | 3g | Activity | = | 2 | % | ALA926597 | % | Homo sapiens | |||
17. | ALA251921 | 4b | Activity | = | 0 | % | ALA926597 | % | Homo sapiens | |||
18. | ALA400943 | 4c | Activity | = | 2 | % | ALA926597 | % | Homo sapiens | |||
19. | ALA251932 | 4d | Activity | = | 3 | % | ALA926597 | % | Homo sapiens | |||
20. | ALA253156 | 4e | Activity | = | 17 | % | ALA926597 | % | Homo sapiens |