# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 2-Arachidonoyl glycerol-d8 | 2-AG | Ki | = | 472 | nM | ALA3782513 | 6.33 | nM | Rattus norvegicus | ||
2. | Arachidonylethanolamide | Table 1 | Ki | = | 89 | nM | ALA3782513 | 7.05 | nM | Rattus norvegicus | ||
3. | δ⁹-tetrahydrocannabinol | 3 | Ki | = | 36 | nM | ALA3782512 | 7.44 | nM | Rattus norvegicus | ||
4. | AM251 | 4 | INH | = | 38 | % | ALA3614948 | % | Rattus norvegicus | |||
5. | ALA3613003 | 52, JZP-169 | INH | = | 104 | % | ALA3614947 | % | Rattus norvegicus | |||
6. | HU 210 | 4 | Activity | = | 306 | % | ALA3614943 | % | Rattus norvegicus | |||
7. | ALA3613003 | 52, JZP-169 | Activity | = | 96 | % | ALA3614942 | % | Rattus norvegicus | |||
8. | ALA5266282 | 18 | Ki | = | 145 | nM | ALA5245485 | 6.84 | nM | Rattus norvegicus | ||
9. | Cannabidiol | 3 | Ki | > | 10 | uM | ALA5245484 | nM | Rattus norvegicus | |||
10. | ALA5282889 | 76 | EC50 | = | 13.3 | nM | ALA5244755 | 7.88 | nM | Rattus norvegicus | ||
11. | ALA5269105 | 3; HU-308 | Ki | > | 10000 | nM | ALA5231891 | nM | Rattus norvegicus | |||
12. | ALA5285808 | 2; JWH-133 | Ki | = | 677 | nM | ALA5231888 | 6.17 | nM | Rattus norvegicus | ||
13. | ALA5281620 | 1; JWH-139 | Ki | = | 2290 | nM | ALA5231888 | 5.64 | nM | Rattus norvegicus | ||
14. | HU-308 | HU308 | Ki | > | 10 | uM | ALA5224282 | nM | Rattus norvegicus | |||
15. | ALA286222 | 15 | Ki | = | 23 | nM | ALA5224276 | 7.64 | nM | Rattus norvegicus | ||
16. | Rimonabant | 4 | Ki | = | 11.5 | nM | ALA5224273 | 7.94 | nM | Rattus norvegicus | ||
17. | AM251 | 4 | Ki | = | 2290 | nM | ALA5224273 | 5.64 | nM | Rattus norvegicus | ||
18. | AM251 | 4 | Ki | = | 7.49 | nM | ALA5224273 | 8.13 | nM | Rattus norvegicus | ||
19. | ALA5183405 | 41c; AM8941 | Emax | = | 97 | % | ALA5157808 | % | Rattus norvegicus | |||
20. | ALA5176554 | 35c; AM8904 | Emax | = | 108 | % | ALA5157808 | % | Rattus norvegicus |