# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PU 02 | SID24807873 | IC50 | = | 0.43 | uM | ALA4219556 | 6.37 | nM | Homo sapiens | ||
2. | VUF 10166 | 26 | Ki | = | 22 | nM | ALA4219561 | 7.66 | nM | Homo sapiens | ||
3. | [³H]meta-chlorophenylbiguanide | 2 (mCPBG) | EC50 | = | 2.8 | uM | ALA4219563 | 5.55 | nM | Homo sapiens | ||
4. | Palonosetron | Palonosetron | Kd | = | 0.18 | nM | ALA3094576 | 9.74 | nM | Homo sapiens | ||
5. | Palonosetron | Palonosetron | IC50 | = | 0.88 | nM | ALA3097163 | 9.06 | nM | Homo sapiens | ||
6. | ALA289469 | 1 | Kd | = | 0.2 | nM | ALA3094576 | 9.70 | nM | Homo sapiens | ||
7. | ALA289469 | 1 | EC50 | = | 0.5 | uM | ALA3097183 | 6.30 | nM | Homo sapiens |