| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5201248 | 38 | INH | = | 26 | % | ALA5157181 | % | Homo sapiens | |||
| 2. |  ALA4567486 | ZG02 | Activity | = | 362 | nM | ALA4409758 | nM | Homo sapiens | |||
| 3. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405639 | % | Homo sapiens | |||
| 4. |  Prexasertib | PREXASERTIB | IC50 | = | 101.62 | nM | ALA4394700 | 6.99 | nM | Homo sapiens | ||
| 5. |  ALA4577258 | (R)-17Ac | IC50 | = | 107.5 | nM | ALA4394700 | 6.97 | nM | Homo sapiens | ||
| 6. |  ALA4749965 | Example 32 | INH | 0 | ALA4739722 | Not Active | % | Homo sapiens | ||||
| 7. |  ALA4537786 | 1g | pEC50 | 0 | ALA4350313 | Not Active | Homo sapiens | |||||
| 8. |  ALA4537753 | 3b | pEC50 | = | 6.35 | ALA4350313 | 6.35 | nM | Homo sapiens | |||
| 9. |  ALA4466855 | 2b | pEC50 | = | 6.47 | ALA4350313 | 6.47 | nM | Homo sapiens | |||
| 10. |  ALA4469542 | 1b | pEC50 | = | 4.6 | ALA4350313 | 4.60 | nM | Homo sapiens | |||
| 11. | ALA4537753 | 3b | FC | = | 4 | ALA4350322 | Homo sapiens | |||||
| 12. | ALA4466855 | 2b | FC | = | 2.81 | ALA4350322 | Homo sapiens | |||||
| 13. | ALA4537786 | 1g | FC | 0 | ALA4350322 | Not Active | Homo sapiens | |||||
| 14. | ALA4469542 | 1b | FC | = | 1.56 | ALA4350322 | Homo sapiens | |||||
| 15. |  2-((2-(2-Bromo-4-methylphenoxy)ethyl)thio)pyrimidine | ZLN-024 | EC50 | = | 0.55 | uM | ALA4350313 | 6.26 | nM | Homo sapiens | ||
| 16. | ALA4537753 | 3b | EC50 | = | 0.44 | uM | ALA4350313 | 6.36 | nM | Homo sapiens | ||
| 17. | ALA4466855 | 2b | EC50 | = | 0.34 | uM | ALA4350313 | 6.47 | nM | Homo sapiens | ||
| 18. | ALA4469542 | 1b | EC50 | = | 109 | uM | ALA4350313 | nM | Homo sapiens | |||
| 19. | 2-((2-(2-Bromo-4-methylphenoxy)ethyl)thio)pyrimidine | ZLN-024 | Activity | = | 156.8 | % | ALA4350309 | % | Homo sapiens | |||
| 20. |  ALA4587164 | 3d | Activity | = | -36.4 | % | ALA4350309 | % | Homo sapiens |
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