# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3754234 | JS1 | Stability | > | 90 | % | ALA3755120 | % | Homo sapiens | |||
2. | Lys-(des-Arg9, Leu8)-Bradykinin trifluoroacetate salt | KL | Stability | 0 | ALA3755112 | Unstable | % | Homo sapiens | ||||
3. | ALA3753868 | RV | Stability | 0 | ALA3755112 | Unstable | % | Homo sapiens | ||||
4. | ALA4172319 | 3 | Ki(app) | = | 294 | uM | ALA4140928 | nM | Homo sapiens | |||
5. | ALA4167456 | 11 | Ki(app) | = | 56 | uM | ALA4140928 | 4.25 | nM | Homo sapiens | ||
6. | ALA4165424 | 19 | Ki(app) | = | 413 | uM | ALA4140928 | nM | Homo sapiens | |||
7. | ALA4173339 | 20 | Ki(app) | = | 289 | uM | ALA4140928 | nM | Homo sapiens | |||
8. | ALA4168849 | 21 | Ki(app) | = | 238 | uM | ALA4140928 | nM | Homo sapiens | |||
9. | ALA4176703 | 22 | Ki(app) | = | 60.4 | uM | ALA4140928 | 4.22 | nM | Homo sapiens | ||
10. | ALA4172319 | 3 | Kinact | = | 0.82 | /min | ALA4140928 | /min | Homo sapiens | |||
11. | ALA4167456 | 11 | Kinact | = | 0.52 | /min | ALA4140928 | /min | Homo sapiens | |||
12. | ALA4165424 | 19 | Kinact | = | 0.6 | /min | ALA4140928 | /min | Homo sapiens | |||
13. | ALA4173339 | 20 | Kinact | = | 0.69 | /min | ALA4140928 | /min | Homo sapiens | |||
14. | ALA4168849 | 21 | Kinact | = | 0.71 | /min | ALA4140928 | /min | Homo sapiens | |||
15. | ALA4176703 | 22 | Kinact | = | 0.47 | /min | ALA4140928 | /min | Homo sapiens | |||
16. | ALA368684 | tableII | IC50 | = | 3.9 | uM | ALA3580144 | 5.41 | nM | Homo sapiens | ||
17. | ALA175436 | tableII | IC50 | = | 1.1 | uM | ALA3580144 | 5.96 | nM | Homo sapiens | ||
18. | ALA3577334 | 1c | IC50 | > | 100 | uM | ALA3580144 | nM | Homo sapiens | |||
19. | ALA446236 | 4 | IC50 | 0 | ALA3580144 | Not Determined | Homo sapiens | |||||
20. | ALA4460840 | 1 | Ki | = | 0.04 | nM | ALA4413958 | 10.40 | nM | Homo sapiens |