# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5220960 | 34 | Ratio IC50 | > | 810 | ALA5217728 | Homo sapiens | |||||
2. | Odanacatib (MK-0822) | 24, odanacatib | Ratio IC50 | < | 300 | ALA5217728 | Homo sapiens | |||||
3. | ALA4763197 | 12 | Ratio Ki | = | 5.8 | ALA4727791 | Homo sapiens | |||||
4. | ALA4788237 | 24 | Ratio Ki | > | 30 | ALA4727791 | Homo sapiens | |||||
5. | ALA4742887 | 7o | Ratio pKi | > | 50 | ALA4678410 | Homo sapiens | |||||
6. | (1R,2R)-N-(1-cyanocyclopropyl)-2-[4-[4-(1,1-dioxo-1,4-thiazinan-4-yl)phenyl]-2-(4-fluorophenyl)-1,3-oxazol-5-yl]cyclohexane-1-carboxamide | 23 | Ratio IC50 | > | 20000 | ALA5106298 | Homo sapiens | |||||
7. | ALA523352 | (R,R)-31 | Ratio IC50 | = | 1355 | ALA5106298 | Homo sapiens | |||||
8. | ALA218007 | 17h | Ratio IC50 | = | 300 | ALA911399 | Homo sapiens | |||||
9. | ALA449096 | 17g | Ratio IC50 | = | 770 | ALA911399 | Homo sapiens | |||||
10. | ALA3085035 | 11e | Selectivity ratio | > | 1000 | ALA911212 | Homo sapiens | |||||
11. | ALA214591 | 10 | Selectivity ratio | > | 1000 | ALA910889 | Homo sapiens | |||||
12. | ALA184514 | 44(R)-2 | Selectivity ratio | = | 212 | ALA866107 | Homo sapiens | |||||
13. | ALA213244 | 16 | Selectivity ratio | = | 1200 | ALA866107 | Homo sapiens | |||||
14. | ALA213194 | 15 | Selectivity ratio | = | 1541 | ALA866107 | Homo sapiens | |||||
15. | ALA212879 | 14 | Selectivity ratio | = | 4307 | ALA866107 | Homo sapiens | |||||
16. | ALA211737 | 13 | Selectivity ratio | = | 2714 | ALA866107 | Homo sapiens | |||||
17. | ALA212907 | 12 | Selectivity ratio | = | 7000 | ALA866107 | Homo sapiens | |||||
18. | ALA213930 | 11 | Selectivity ratio | = | 1384 | ALA866107 | Homo sapiens | |||||
19. | ALA202554 | 25d | Selectivity ratio | 0 | ALA864078 | Not Determined | Homo sapiens | |||||
20. | ALA201733 | 25c | Selectivity ratio | 0 | ALA864078 | Not Determined | Homo sapiens |