| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2364562 | 8a | Km | = | 110 | nM | ALA869161 | nM | Homo sapiens | |||
| 2. |  β-Nicotinamide adenine dinucleotide hydrate | NAD | Km | = | 100 | uM | ALA869161 | nM | Homo sapiens | |||
| 3. |  Mycophenolic acid | MPA | Selectivity ratio | = | 2.9 | ALA865553 | Homo sapiens | |||||
| 4. |  ALA428633 | 25 | Selectivity ratio | = | 3.6 | ALA865553 | Homo sapiens | |||||
| 5. |  ALA209069 | 26 | Selectivity ratio | = | 1.7 | ALA865553 | Homo sapiens | |||||
| 6. |  ALA208921 | 27 | Selectivity ratio | = | 2.8 | ALA865553 | Homo sapiens | |||||
| 7. |  ALA610157 | 5 | Ki | = | 600 | uM | ALA697164 | nM | Homo sapiens | |||
| 8. |  ALA610153 | 4 | Ki | = | 46 | uM | ALA697164 | 4.34 | nM | Homo sapiens | ||
| 9. |  Inosine 5'-Monophosphate(IMP) | IMPs from Table 3 | Km | = | 12 | uM | ALA697165 | nM | Homo sapiens | |||
| 10. |  ALA609835 | 6 | Ki | = | 190 | uM | ALA697164 | nM | Homo sapiens | |||
| 11. |  ALA611590 | 2 | Ki | = | 120 | uM | ALA697164 | nM | Homo sapiens | |||
| 12. |  ALA1242996 | GMP | Ki | = | 38 | uM | ALA697164 | 4.42 | nM | Homo sapiens | ||
| 13. |  ALA1683023 | 6-chloropurine ribonucleoside monophosphate | K inact | = | 0.076 | M-1 min-1 | ALA697167 | M-1 min-1 | Homo sapiens | |||
| 14. | ALA1683023 | 6-chloropurine ribonucleoside monophosphate | Ki | = | 62 | uM | ALA697166 | 4.21 | nM | Homo sapiens | ||
| 15. |  ALA607780 | FVIMP(2-[2-(Z)-fluroviny]inosine 5'-monophosphate) | K inact | = | 0.027 | s-1 | ALA697167 | s-1 | Homo sapiens | |||
| 16. | ALA607780 | FVIMP(2-[2-(Z)-fluroviny]inosine 5'-monophosphate) | Ki | = | 1.11 | uM | ALA697166 | 5.96 | nM | Homo sapiens | ||
| 17. |  ALA45771 | 14 | IC50 | = | 8.1 | uM | ALA699983 | 5.09 | nM | Homo sapiens | ||
| 18. |  ALA47067 | 13 | IC50 | = | 4.4 | uM | ALA699983 | 5.36 | nM | Homo sapiens | ||
| 19. |  4-Hydroxycarbazole | MFCD02178385 | IC50 | = | 54 | uM | ALA699983 | 4.27 | nM | Homo sapiens | ||
| 20. |  ALA23526 | Thiophenthiofurin | Inhibition | = | 83.2 | % | ALA697168 | % | Homo sapiens |
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