# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | JWH-018 | 3, JWH-018 | Emax | = | 167 | % | ALA4360759 | % | Rattus norvegicus | |||
2. | JWH-018 | 3, JWH-018 | EC50 | = | 36 | nM | ALA4360757 | 7.44 | nM | Rattus norvegicus | ||
3. | AM-630 | AM-630 | Emax | = | 100 | % | ALA4360753 | % | Rattus norvegicus | |||
4. | Rimonabant | 4 | Emax | = | 100 | % | ALA4360753 | % | Rattus norvegicus | |||
5. | ALA4441099 | 12 | Emax | = | 110 | % | ALA4360753 | % | Rattus norvegicus | |||
6. | ALA4526969 | 10 | Emax | = | 107 | % | ALA4360753 | % | Rattus norvegicus | |||
7. | Endomorphin 2 TFA | 1 | Activity | 0 | ALA4360739 | Not Active | Rattus norvegicus | |||||
8. | Endomorphin 1 | 1 | Activity | 0 | ALA4360739 | Not Active | Rattus norvegicus | |||||
9. | [³H]naloxone | naloxone | Activity | 0 | ALA4360739 | Not Active | Rattus norvegicus | |||||
10. | morphine | morphine | Activity | 0 | ALA4360739 | Not Active | Rattus norvegicus | |||||
11. | JWH-018 | 3, JWH-018 | Kd(app) | = | 6.5 | nM | ALA4360717 | 8.19 | nM | Rattus norvegicus | ||
12. | JWH-018 | 3, JWH-018 | Emax | = | 1120 | fmol/mg | ALA4360749 | fmol/mg | Rattus norvegicus | |||
13. | JWH-018 | 3, JWH-018 | Kdiss | = | 0.105 | /min | ALA4360717 | /min | Rattus norvegicus | |||
14. | ALA4572221 | 21 | Ki | = | 1042 | nM | ALA4360730 | 5.98 | nM | Rattus norvegicus | ||
15. | ALA4533639 | 20 | Ki | = | 1216 | nM | ALA4360730 | 5.92 | nM | Rattus norvegicus | ||
16. | ALA4575678 | 19 | Ki | = | 317 | nM | ALA4360730 | 6.50 | nM | Rattus norvegicus | ||
17. | ALA4456884 | 18 | Ki | = | 823 | nM | ALA4360730 | 6.08 | nM | Rattus norvegicus | ||
18. | ALA4557161 | 17 | Ki | = | 149 | nM | ALA4360730 | 6.83 | nM | Rattus norvegicus | ||
19. | ALA4443479 | 16 | Ki | = | 269 | nM | ALA4360730 | 6.57 | nM | Rattus norvegicus | ||
20. | ALA235743 | YDAGF-NH2 | Ki | > | 10000 | nM | ALA4360730 | nM | Rattus norvegicus |