# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3924528 | BDBM245222 | INH | 0 | ALA5140275 | Active | % | Homo sapiens | ||||
2. | ALA4758056 | TD-004 | INH | = | 90 | % | ALA5137681 | % | Homo sapiens | |||
3. | ALA3734798 | 3 | IC50 | = | 64 | nM | ALA4716886 | 7.19 | nM | Homo sapiens | ||
4. | ALA4762256 | 12a | IC50 | = | 3 | nM | ALA4716886 | 8.52 | nM | Homo sapiens | ||
5. | ALA4780490 | 16a | IC50 | = | 328 | nM | ALA4716886 | 6.48 | nM | Homo sapiens | ||
6. | ALA4762861 | 20a | IC50 | = | 7 | nM | ALA4716886 | 8.15 | nM | Homo sapiens | ||
7. | ALA3651854 | BDBM107057 | IC50 | = | 26 | nM | ALA4716886 | 7.58 | nM | Homo sapiens | ||
8. | ALA4787280 | 26 | IC50 | = | 7310 | nM | ALA4716886 | 5.14 | nM | Homo sapiens | ||
9. | ALA4739938 | 27 | IC50 | = | 2867 | nM | ALA4716886 | 5.54 | nM | Homo sapiens | ||
10. | ALA4762929 | 30b | IC50 | = | 1344 | nM | ALA4716886 | 5.87 | nM | Homo sapiens | ||
11. | ALA4795530 | 32 | IC50 | = | 6851 | nM | ALA4716886 | 5.16 | nM | Homo sapiens | ||
12. | ALA3651854 | BDBM107057 | IC50 | = | 0.03 | uM | ALA4716831 | 7.52 | nM | Homo sapiens | ||
13. | LDK378 | 6, LDK378 | IC50 | = | 26 | nM | ALA4716830 | 7.58 | nM | Homo sapiens | ||
14. | ALA3734798 | 3 | IC50 | = | 151 | nM | ALA4716830 | 6.82 | nM | Homo sapiens | ||
15. | ALA4779222 | 11a | IC50 | = | 47 | nM | ALA4716830 | 7.33 | nM | Homo sapiens | ||
16. | ALA4791252 | 11d | IC50 | = | 33 | nM | ALA4716830 | 7.48 | nM | Homo sapiens | ||
17. | ALA4762256 | 12a | IC50 | = | 6 | nM | ALA4716830 | 8.22 | nM | Homo sapiens | ||
18. | ALA4798141 | 12d | IC50 | = | 13 | nM | ALA4716830 | 7.89 | nM | Homo sapiens | ||
19. | ALA3651885 | BDBM107097 | IC50 | = | 47 | nM | ALA4716830 | 7.33 | nM | Homo sapiens | ||
20. | ALA4780490 | 16a | IC50 | = | 684 | nM | ALA4716830 | 6.17 | nM | Homo sapiens |