# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2152768 | 3 | INH | = | -1.1 | % | ALA2156499 | % | Homo sapiens | |||
2. | ALA3125728 | 18 | Activity | = | 95 | % | ALA3132650 | % | Homo sapiens | |||
3. | ALA3125726 | 20 | Activity | = | 103 | % | ALA3132650 | % | Homo sapiens | |||
4. | ALA3125727 | 19 | Activity | = | 100 | % | ALA3132650 | % | Homo sapiens | |||
5. | ALA2180408 | Figure 27, R1C1 | % inhibition | -1 | % | ALA4886208 | Not Active | % | Homo sapiens | |||
6. | ALA4475494 | 19 | % Inhibition | 2.5 | % | ALA4885929 | Not Active | % | Homo sapiens | |||
7. | ALA4580220 | EUB0000311 | % residual kinase activity | 91 | % | ALA4884255 | Not Active | % | Homo sapiens | |||
8. | CLK-IN-T3 | EUB0000321 | % inhibition | -13.964 | % | ALA4883278 | Not Active | % | Homo sapiens | |||
9. | CLK-IN-T3 | EUB0000321 | % inhibition | -16.992 | % | ALA4883278 | Not Active | % | Homo sapiens | |||
10. | MLI-2 | 1; MLi-2 | % Inhibition | 11.329 | % | ALA4882686 | Not Active | % | Homo sapiens | |||
11. | BAY-885 | BAY-885; 41 | % residual kinase activity | 103 | % | ALA4880991 | Not Active | % | Homo sapiens | |||
12. | 2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | % inhibition | -10 | % | ALA4880590 | Not Active | % | Homo sapiens | |||
13. | ALA3297832 | 4 | IC50 | = | 0.82 | uM | ALA3299307 | 6.09 | nM | Homo sapiens | ||
14. | ALA3289600 | 5e | IC50 | > | 10 | uM | ALA3293378 | nM | Homo sapiens | |||
15. | ALA3289596 | 5a | IC50 | > | 10 | uM | ALA3293378 | nM | Homo sapiens | |||
16. | ALA3421644 | 7t | IC50 | = | 0.3 | uM | ALA3424710 | 6.52 | nM | Homo sapiens | ||
17. | ALA3422750 | 7o | IC50 | = | 5.6 | uM | ALA3424710 | 5.25 | nM | Homo sapiens | ||
18. | ALA3422748 | 7m | IC50 | = | 1.9 | uM | ALA3424710 | 5.72 | nM | Homo sapiens | ||
19. | ALA3422747 | 7l | IC50 | = | 0.4 | uM | ALA3424710 | 6.40 | nM | Homo sapiens | ||
20. | ALA3422744 | 7i | IC50 | = | 0.7 | uM | ALA3424710 | 6.16 | nM | Homo sapiens |