# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (1R,2R)-N-(1-cyanocyclopropyl)-2-[4-[4-(1,1-dioxo-1,4-thiazinan-4-yl)phenyl]-2-(4-fluorophenyl)-1,3-oxazol-5-yl]cyclohexane-1-carboxamide | 23 | Ratio IC50 | > | 20000 | ALA5106297 | Homo sapiens | |||||
2. | ALA523352 | (R,R)-31 | Ratio IC50 | = | 5556 | ALA5106297 | Homo sapiens | |||||
3. | ALA5220960 | 34 | Ratio IC50 | > | 1620 | ALA5217729 | Homo sapiens | |||||
4. | Odanacatib (MK-0822) | 24, odanacatib | Ratio IC50 | < | 1180 | ALA5217729 | Homo sapiens | |||||
5. | ALA184514 | 44(R)-2 | Selectivity ratio | = | 481 | ALA866106 | Homo sapiens | |||||
6. | ALA213244 | 16 | Selectivity ratio | = | 17000 | ALA866106 | Homo sapiens | |||||
7. | ALA213194 | 15 | Selectivity ratio | = | 10625 | ALA866106 | Homo sapiens | |||||
8. | ALA212879 | 14 | Selectivity ratio | = | 28461 | ALA866106 | Homo sapiens | |||||
9. | ALA211737 | 13 | Selectivity ratio | = | 3428 | ALA866106 | Homo sapiens | |||||
10. | ALA212907 | 12 | Selectivity ratio | = | 22500 | ALA866106 | Homo sapiens | |||||
11. | ALA213930 | 11 | Selectivity ratio | = | 16923 | ALA866106 | Homo sapiens | |||||
12. | ALA202554 | 25d | Selectivity ratio | 0 | ALA864077 | Not Determined | Homo sapiens | |||||
13. | ALA201733 | 25c | Selectivity ratio | 0 | ALA864077 | Not Determined | Homo sapiens | |||||
14. | ALA381135 | 25b | Selectivity ratio | 0 | ALA864077 | Not Determined | Homo sapiens | |||||
15. | ALA427377 | 25a | Selectivity ratio | 0 | ALA864077 | Not Determined | Homo sapiens | |||||
16. | ALA439517 | 2c | Ratio IC50 | = | 7100 | ALA866590 | Homo sapiens | |||||
17. | ALA204284 | 2d | Ratio IC50 | = | 4300 | ALA866590 | Homo sapiens | |||||
18. | ALA206482 | 2f | Ratio IC50 | = | 2900 | ALA866590 | Homo sapiens | |||||
19. | ALA203027 | 2g | Ratio IC50 | = | 5200 | ALA866590 | Homo sapiens | |||||
20. | ALA383238 | 2h | Ratio IC50 | > | 10000 | ALA866590 | Homo sapiens |