# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tubastatin A | Tubastatin A | IC50 | > | 30 | uM | ALA2432125 | nM | Homo sapiens | |||
2. | Tubacin | Tubacin | IC50 | = | 1.27 | uM | ALA2432125 | 5.90 | nM | Homo sapiens | ||
3. | Tubacin | Tubacin | IC50 | = | 1.27 | uM | ALA2424317 | 5.90 | nM | Homo sapiens | ||
4. | Tubastatin A | Tubastatin A | IC50 | > | 30 | uM | ALA2424317 | nM | Homo sapiens | |||
5. | ALA99 | TSA | Activity | = | 0.95 | % | ALA2399517 | % | Homo sapiens | |||
6. | ALA2398525 | 39 | Activity | = | 53.2 | % | ALA2399517 | % | Homo sapiens | |||
7. | ALA2398523 | 37 | Activity | > | 75 | % | ALA2399517 | % | Homo sapiens | |||
8. | ALA2398524 | 38 | Activity | > | 75 | % | ALA2399517 | % | Homo sapiens | |||
9. | ALA2063397 | 27 | INH | 0 | ALA2065959 | Active | % | Homo sapiens | ||||
10. | ALA2063396 | 26 | Ki | = | 37 | nM | ALA2065957 | 7.43 | nM | Homo sapiens | ||
11. | ALA2063396 | 26 | INH | = | 60 | % | ALA2065939 | % | Homo sapiens | |||
12. | ALA2063395 | 15 | IC50 | = | 1.4 | uM | ALA2065942 | 5.85 | nM | Homo sapiens | ||
13. | ALA2063396 | 26 | IC50 | = | 0.8 | uM | ALA2065942 | 6.10 | nM | Homo sapiens | ||
14. | Vorinostat (SAHA, MK0683) | SAHA | IC50 | = | 0.043 | uM | ALA2065942 | 7.37 | nM | Homo sapiens | ||
15. | Romidepsin (FK228, Depsipeptide) | FK-228 | IC50 | = | 3 | nM | ALA2065942 | 8.52 | nM | Homo sapiens | ||
16. | ALA2063396 | 26 | Ratio IC50 | = | 40 | ALA2065946 | Homo sapiens | |||||
17. | Vorinostat (SAHA, MK0683) | SAHA | IC50 | = | 41 | nM | ALA2014771 | 7.39 | nM | Homo sapiens | ||
18. | ALA430060 | 1 | IC50 | = | 29 | nM | ALA2014771 | 7.54 | nM | Homo sapiens | ||
19. | ALA2012818 | 19 | IC50 | = | 16 | nM | ALA2014771 | 7.80 | nM | Homo sapiens | ||
20. | ALA2012817 | 18 | IC50 | = | 9 | nM | ALA2014771 | 8.05 | nM | Homo sapiens |