# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GW841819X | 1, GW841819X | Kd | > | 50 | uM | ALA2156122 | nM | Homo sapiens | |||
2. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886878 | nM | Homo sapiens | |||||
3. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886823 | nM | Homo sapiens | ||||
4. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885820 | nM | Homo sapiens | |||||
5. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885760 | nM | Homo sapiens | ||||
6. | ALA4648362 | EUB0001116 | pKd | 4.8 | ALA4885696 | nM | Homo sapiens | |||||
7. | ALA3356574 | 5 | Kd | = | 350 | uM | ALA3430213 | 3.46 | nM | Homo sapiens | ||
8. | ALA3410003 | 40a | deltaTm | = | 3.55 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
9. | ALA3410002 | 39b | deltaTm | = | 2.7 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
10. | ALA3410000 | 33b | deltaTm | = | 3.42 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
11. | ALA3409996 | 25 | deltaTm | = | 3.28 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
12. | ALA3409993 | 18b | deltaTm | = | 1.36 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
13. | ALA3409992 | 18a | deltaTm | = | 1.44 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
14. | (+)-JQ1 | (+)-JQ1 | deltaTm | = | 1.04 | degrees C | ALA3414215 | degrees C | Homo sapiens | |||
15. | ALA3356579 | 12 | Kd | = | 500 | uM | ALA3380074 | 3.30 | nM | Homo sapiens | ||
16. | ALA3356578 | 11 | Kd | = | 500 | uM | ALA3380074 | 3.30 | nM | Homo sapiens | ||
17. | ALA3356577 | 10 | Kd | = | 450 | uM | ALA3380074 | 3.35 | nM | Homo sapiens | ||
18. | ALA1338624 | SID845570 | Kd | = | 400 | uM | ALA3380074 | 3.40 | nM | Homo sapiens | ||
19. | ALA3356576 | 8 | Kd | = | 600 | uM | ALA3380074 | 3.22 | nM | Homo sapiens | ||
20. | ALA3356575 | 7 | Kd | = | 450 | uM | ALA3380074 | 3.35 | nM | Homo sapiens |