# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK8814 | 32 | pIC50 | = | 7.3 | ALA5232451 | 7.30 | nM | Homo sapiens | |||
2. | ALA5279678 | 39 | Kd | = | 2.4 | mM | ALA5232450 | 2.62 | nM | Homo sapiens | ||
3. | ALA5286790 | 10 | IC50 | = | 55 | uM | ALA5225193 | 4.26 | nM | Homo sapiens | ||
4. | ALA5285969 | 9 | IC50 | = | 543 | uM | ALA5225193 | nM | Homo sapiens | |||
5. | ALA5274345 | 8 | IC50 | = | 822 | uM | ALA5225193 | nM | Homo sapiens | |||
6. | ALA5284806 | FL33 | IC50 | = | 377 | uM | ALA5225193 | nM | Homo sapiens | |||
7. | ALA4451357 | 19 | Activity | = | 70 | % | ALA4415512 | % | Homo sapiens | |||
8. | BAY-850 | 4; BAY-850 | IC50 | = | 166 | nM | ALA4382889 | 6.78 | nM | Homo sapiens | ||
9. | ALA4648362 | EUB0001116 | pKd | = | 4.8 | ALA4727063 | 4.80 | nM | Homo sapiens | |||
10. | ALA4785142 | 18, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
11. | ALA4785133 | 17, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
12. | ALA4745677 | 16, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
13. | ALA4752082 | 15, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
14. | ALA4781414 | 14, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
15. | ALA4796868 | 13, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
16. | ALA4760227 | 12, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
17. | ALA4765129 | 11, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
18. | ALA4746291 | 10, Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
19. | ALA4778637 | 9, Cis isomer | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens | ||||
20. | ALA4787240 | 8, rac-Mixture of trans (1:1) | pIC50 | < | 4.4 | ALA4727046 | nM | Homo sapiens |