# | Name | Compound Key | Action Type | Relation | Activety Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1725922 | SID24397477 | IC50 | = | 5.6 | uM | ALA2168840 | 5.25 | nM | Mus musculus | ||
2. | 10-(4-ethylphenyl)sulfonyl-N-(thiophen-2-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine | SID24397505 | IC50 | = | 11 | nM | ALA2168840 | 7.96 | nM | Mus musculus | ||
3. | ALA2165789 | 2az | IC50 | > | 25 | uM | ALA2168840 | nM | Mus musculus | |||
4. | ALA1173569 | 2{3,7} | IC50 | = | 212 | nM | ALA2168840 | 6.67 | nM | Mus musculus | ||
5. | ALA1372659 | SID24397449 | IC50 | = | 153 | nM | ALA2168840 | 6.82 | nM | Mus musculus | ||
6. | ALA2165780 | 3b | IC50 | = | 16500 | nM | ALA2168840 | 4.78 | nM | Mus musculus | ||
7. | ALA2165781 | 3c | IC50 | = | 537 | nM | ALA2168840 | 6.27 | nM | Mus musculus | ||
8. | ALA2165782 | 3d | IC50 | = | 1110 | nM | ALA2168840 | 5.96 | nM | Mus musculus | ||
9. | ALA2165783 | 3e | IC50 | = | 5290 | nM | ALA2168840 | 5.28 | nM | Mus musculus | ||
10. | ALA2165784 | 3f | IC50 | = | 104 | nM | ALA2168840 | 6.98 | nM | Mus musculus | ||
11. | ALA2165785 | 3g | IC50 | = | 196 | nM | ALA2168840 | 6.71 | nM | Mus musculus | ||
12. | ALA2165786 | 3h | IC50 | = | 468 | nM | ALA2168840 | 6.33 | nM | Mus musculus | ||
13. | ALA1590659 | SID24397607 | IC50 | = | 32 | nM | ALA2168840 | 7.50 | nM | Mus musculus | ||
14. | ALA2165787 | 3j | IC50 | > | 2500 | nM | ALA2168840 | nM | Mus musculus | |||
15. | ALA2165788 | 3k | IC50 | = | 14 | nM | ALA2168840 | 7.85 | nM | Mus musculus | ||
16. | 10-(4-ethylphenyl)sulfonyl-N-(thiophen-2-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine | SID24397505 | IC50 | = | 25.1 | nM | ALA2167858 | 7.60 | nM | Mus musculus | ||
17. | ALA2165788 | 3k | IC50 | = | 23 | nM | ALA2167856 | 7.64 | nM | Mus musculus | ||
18. | ALA2165788 | 3k | INH | 0 | ALA2167856 | Dose-dependent effect | % | Mus musculus | ||||
19. | ALA5087071 | 26 | IC50 | = | 0.16 | uM | ALA5033690 | 6.80 | nM | Mus musculus | ||
20. | ALA5091857 | 25e | IC50 | > | 10 | uM | ALA5033690 | nM | Mus musculus |