# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5190238 | (1R,5S,8S)-5a | Activity | = | 0 | % | ALA5157656 | % | Rattus norvegicus | |||
2. | ALA5203422 | (1S,5R,8R)-5a | Activity | = | 0 | % | ALA5157656 | % | Rattus norvegicus | |||
3. | ALA5204863 | (1R,5R,7S)-4b | Activity | = | 0 | % | ALA5157656 | % | Rattus norvegicus | |||
4. | ALA5178401 | (1S,5S,7R)-4b | Activity | = | 0 | % | ALA5157656 | % | Rattus norvegicus | |||
5. | ALA5185196 | (1R,5R,7S)-4a | Activity | = | 0 | % | ALA5157656 | % | Rattus norvegicus | |||
6. | SNC80 | SNC-80 | Ki | = | 1.2 | nM | ALA5157651 | 8.92 | nM | Rattus norvegicus | ||
7. | Naloxone | naloxone | Ki | = | 103 | nM | ALA5157651 | 6.99 | nM | Rattus norvegicus | ||
8. | ALA5200121 | rac-5b | Ki | > | 1000 | nM | ALA5157651 | nM | Rattus norvegicus | |||
9. | ALA5173028 | (1S,5S,7R)-4a | Ki | = | 542 | nM | ALA5157651 | 6.27 | nM | Rattus norvegicus | ||
10. | ALA5202222 | 5e | Emax | = | 209.8 | % | ALA5141740 | % | Rattus norvegicus | |||
11. | ALA5206165 | 5d | Emax | = | 205.5 | % | ALA5141740 | % | Rattus norvegicus | |||
12. | ALA5180450 | 5a | Emax | = | 158.1 | % | ALA5141740 | % | Rattus norvegicus | |||
13. | ALA5178795 | 4a; SLL-627 | Emax | = | 193.9 | % | ALA5141740 | % | Rattus norvegicus | |||
14. | ALA5200910 | 3 | Emax | = | 186.4 | % | ALA5141740 | % | Rattus norvegicus | |||
15. | ALA5177908 | 2 | Emax | = | 262.5 | % | ALA5141740 | % | Rattus norvegicus | |||
16. | ALA5202222 | 5e | EC50 | = | 1317 | nM | ALA5141739 | 5.88 | nM | Rattus norvegicus | ||
17. | ALA5206165 | 5d | EC50 | = | 950.8 | nM | ALA5141739 | 6.02 | nM | Rattus norvegicus | ||
18. | ALA5178795 | 4a; SLL-627 | EC50 | = | 886.1 | nM | ALA5141739 | 6.05 | nM | Rattus norvegicus | ||
19. | ALA5200910 | 3 | EC50 | = | 43.76 | nM | ALA5141739 | 7.36 | nM | Rattus norvegicus | ||
20. | ALA5177908 | 2 | EC50 | = | 153.5 | nM | ALA5141739 | 6.81 | nM | Rattus norvegicus |