# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886902 | nM | Homo sapiens | |||||
2. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886855 | nM | Homo sapiens | ||||
3. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885852 | nM | Homo sapiens | |||||
4. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885798 | nM | Homo sapiens | ||||
5. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885730 | nM | Homo sapiens | |||||
6. | GSK1324726A (I-BET726) | 45 | pIC50 | = | 4.8 | ALA3383435 | 4.80 | nM | Homo sapiens | |||
7. | GSK1324726A (I-BET726) | 45 | pIC50 | < | 5 | ALA3383434 | nM | Homo sapiens | ||||
8. | OF 1 | 8 | Delta TM | = | -0.23 | C | ALA4650190 | C | Homo sapiens | |||
9. | ALA4650212 | EUB0000324a | Delta TM | = | 0.14 | C | ALA4650190 | C | Homo sapiens | |||
10. | bromosporine | Bromosporine | Delta TM | = | 0.49 | C | ALA4650190 | C | Homo sapiens | |||
11. | OF 1 | 8 | Delta TM | = | -0.61 | C | ALA4650190 | C | Homo sapiens | |||
12. | bromosporine | Bromosporine | Delta TM | = | -0.18 | C | ALA4650190 | C | Homo sapiens | |||
13. | PFI-4 | 11 | Inhibition | = | 35.48 | % | ALA4650040 | % | Homo sapiens | |||
14. | ALA4650212 | EUB0000324a | Inhibition | = | -10.471 | % | ALA4650040 | % | Homo sapiens | |||
15. | OF 1 | 8 | Inhibition | = | 9.058 | % | ALA4650040 | % | Homo sapiens | |||
16. | NI-57 | 76; NI-57 | Inhibition | = | 9.82 | % | ALA4650040 | % | Homo sapiens | |||
17. | bromosporine | Bromosporine | Inhibition | = | 50.425 | % | ALA4650040 | % | Homo sapiens | |||
18. | ALA4852928 | 60; GSK040 | INH | < | 40 | % | ALA4827488 | % | Homo sapiens | |||
19. | ALA4059509 | 36; Nl-198 | IC50 | > | 100000 | nM | ALA4053071 | nM | Homo sapiens | |||
20. | ALA4083840 | 13 | Activity | = | 100 | % | ALA4047559 | % | Homo sapiens |