# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886882 | nM | Homo sapiens | |||||
2. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886827 | nM | Homo sapiens | ||||
3. | GSK620 | 1; 20 | pKd | 4.6 | ALA4885824 | nM | Homo sapiens | |||||
4. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885764 | nM | Homo sapiens | ||||
5. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885700 | nM | Homo sapiens | |||||
6. | ALA5205457 | 3r; ZLD2218 | IC50 | > | 1 | uM | ALA5158668 | nM | Homo sapiens | |||
7. | N-(1,3-dimethyl-2-oxo-6-piperidin-1-ylbenzimidazol-5-yl)-2-methoxybenzamide | SID24270853 | pIC50 | = | 5.1 | ALA3385106 | 5.10 | nM | Homo sapiens | |||
8. | GSK1324726A (I-BET726) | 45 | pIC50 | < | 4.7 | ALA3383437 | nM | Homo sapiens | ||||
9. | ALA2181721 | 6a | deltaTm | < | 1 | degrees C | ALA2186999 | degrees C | Homo sapiens | |||
10. | ALA2181718 | 34 | deltaTm | < | 1 | degrees C | ALA2186999 | degrees C | Homo sapiens | |||
11. | ALA3590408 | 46 | pKi | = | 6.4 | ALA3591380 | 6.40 | nM | Homo sapiens | |||
12. | bromosporine | Bromosporine | Kd | = | 1.653 | uM | ALA4650197 | 5.78 | nM | Homo sapiens | ||
13. | BAZ2-ICR | 13, BAZ2-ICR | Delta TM | = | 0.29 | C | ALA4650062 | C | Homo sapiens | |||
14. | TP-472 | 1; TP-472 | Delta TM | = | 0.25 | C | ALA4650062 | C | Homo sapiens | |||
15. | L-45 | 8; L-Moses | Delta TM | = | -0.26 | C | ALA4650062 | C | Homo sapiens | |||
16. | PFI-4 | 11 | Delta TM | = | 1.99 | C | ALA4650062 | C | Homo sapiens | |||
17. | I-BRD9 | 45; I-BRD9 | Delta TM | = | 0.98 | C | ALA4650062 | C | Homo sapiens | |||
18. | NVS-CECR2-1 | NVS-1 | Delta TM | = | 0.34 | C | ALA4650062 | C | Homo sapiens | |||
19. | ALA4650212 | EUB0000324a | Delta TM | = | 0.01 | C | ALA4650062 | C | Homo sapiens | |||
20. | OF 1 | 8 | Delta TM | = | 3.42 | C | ALA4650062 | C | Homo sapiens |