| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  NI-57 | 76; NI-57 | Kd | = | 110 | nM | ALA3790874 | 6.96 | nM | Homo sapiens | ||
| 2. |  OF-1 | 8 | Kd | = | 500 | nM | ALA3790874 | 6.30 | nM | Homo sapiens | ||
| 3. |  SGC-CBP30 | 72 | deltaTm | = | 2.3 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 4. |  bromosporine | Bromosporine | deltaTm | = | 6.1 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 5. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 1.1 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 6. |  ALA3780429 | 85 | deltaTm | = | 0.1 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 7. |  ALA3779929 | 84 | deltaTm | = | 0.1 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 8. |  ALA3780059 | 73 | deltaTm | = | 1.6 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 9. |  ALA3780128 | 68 | deltaTm | = | 2.9 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 10. |  ALA3781254 | 60 | deltaTm | = | -0.3 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 11. |  ALA3780901 | 58 | deltaTm | = | 0.1 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 12. |  ALA3780381 | 47 | deltaTm | = | 2.1 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 13. |  ALA3234253 | 8e | deltaTm | = | 1.6 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 14. |  N-cyclohexyl-1-ethyl-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide | 28 | deltaTm | = | 2.4 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 15. |  ALA3782048 | 25 | deltaTm | = | 2 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 16. |  ALA3781449 | 20 | deltaTm | = | 1.3 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 17. |  ALA3780398 | 17 | deltaTm | = | 2.9 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 18. |  ALA3780508 | 14 | deltaTm | = | 2 | degrees C | ALA3782669 | degrees C | Homo sapiens | |||
| 19. |  ALA3774575 | 8i; IACS-9571 | Kd | = | 12 | nM | ALA3779322 | 7.92 | nM | Homo sapiens | ||
| 20. |  3,4-dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]benzene-1-sulfonamide | 34 | Kd | = | 1130 | nM | ALA3771493 | 5.95 | nM | Homo sapiens |
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