# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PFI 4 | 11 | pIC50 | = | 4.8 | ALA5214190 | 4.80 | nM | Homo sapiens | |||
2. | PFI 4 | 11 | dTm | = | 2 | K | ALA5214189 | K | Homo sapiens | |||
3. | PFI 4 | 11 | IC50 | = | 3600 | nM | ALA5214188 | 5.44 | nM | Homo sapiens | ||
4. | OF-1 | 8 | dTm | = | 3.1 | K | ALA5214234 | K | Homo sapiens | |||
5. | OF-1 | 8 | IC50 | = | 2200 | nM | ALA5214233 | 5.66 | nM | Homo sapiens | ||
6. | NI-57 | 76; NI-57 | Kd | = | 110 | nM | ALA5214153 | 6.96 | nM | Homo sapiens | ||
7. | NI-57 | 76; NI-57 | IC50 | = | 46 | nM | ALA5214152 | 7.34 | nM | Homo sapiens | ||
8. | GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 110 | nM | ALA5214221 | 6.96 | nM | Homo sapiens | ||
9. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 45 | nM | ALA5214113 | 7.35 | nM | Homo sapiens | ||
10. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 6 | nM | ALA5214112 | 8.22 | nM | Homo sapiens | ||
11. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 97 | nM | ALA5214111 | 7.01 | nM | Homo sapiens | ||
12. | PFI 4 | 11 | Kd | = | 512.86 | nM | ALA5214177 | 6.29 | nM | Homo sapiens | ||
13. | OF-1 | 8 | Kd | = | 505 | nM | ALA5210549 | 6.30 | nM | Homo sapiens | ||
14. | PFI 4 | 11 | Kd | = | 775 | nM | ALA5210542 | 6.11 | nM | Homo sapiens | ||
15. | NI-57 | 76; NI-57 | IC50 | = | 619 | nM | ALA5210535 | 6.21 | nM | Homo sapiens | ||
16. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 67 | nM | ALA5210529 | 7.17 | nM | Homo sapiens | ||
17. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 503 | nM | ALA5210233 | 6.30 | nM | Homo sapiens | ||
18. | OF-1 | 8 | EC50 | > | 500 | nM | ALA5210070 | nM | Homo sapiens | |||
19. | BAY-299 | 5b; atropisomer 2 | GI50 | = | 1060 | nM | ALA5210065 | nM | Homo sapiens | |||
20. | ALA5205457 | 3r; ZLD2218 | IC50 | > | 1 | uM | ALA5158668 | nM | Homo sapiens |