# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886879 | nM | Homo sapiens | |||||
2. | ALA4639128 | 62 | Kd | 25000 | nM | ALA4886824 | nM | Homo sapiens | ||||
3. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885821 | nM | Homo sapiens | |||||
4. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885761 | nM | Homo sapiens | ||||
5. | ALA4648362 | EUB0001116 | pKd | 4.8 | ALA4885697 | nM | Homo sapiens | |||||
6. | GSK1324726A (I-BET726) | 45 | pIC50 | < | 4.5 | ALA3383404 | nM | Homo sapiens | ||||
7. | ALA3590405 | 42 | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
8. | ALA4748520 | H4K5acK12ac (res 1-15) | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
9. | ALA4792431 | H4K5acK8ac (res 1-10) | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
10. | ALA4762063 | H4K12ac (res 4-17) | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
11. | ALA4750026 | H4K5ac (res 1-10) | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
12. | ALA4748867 | H4 unmodified (res 4-17) | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
13. | ALA4751427 | H2AK5ac (res 1-12) | Kd | 0 | ALA4672548 | Not Active | Homo sapiens | |||||
14. | ALA3590405 | 42 | Kd | = | 166.9 | nM | ALA4672541 | 6.78 | nM | Homo sapiens | ||
15. | ALA4781561 | H3K14ac (res 8-19) | Kd | 0 | ALA4672541 | Not Active | Homo sapiens | |||||
16. | ALA4743832 | H3K9ac (res 1-12) | Kd | 0 | ALA4672541 | Not Active | Homo sapiens | |||||
17. | ALA4761046 | H3 unmodified (res 1-12) | Kd | 0 | ALA4672541 | Not Active | Homo sapiens | |||||
18. | ALA4762443 | H4K12acK16ac (res 10-20) | Kd | = | 213.9 | uM | ALA4672541 | nM | Homo sapiens | |||
19. | ALA4748267 | H4K8acK16ac (1-20) | Kd | = | 35.7 | uM | ALA4672541 | 4.45 | nM | Homo sapiens | ||
20. | ALA4757518 | H4K8acK12ac (res 6-15) | Kd | 0 | ALA4672541 | Not Active | Homo sapiens |