# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4532174 | 24 | IC50 | > | 2.5 | uM | ALA5231259 | nM | Homo sapiens | |||
2. | A 366 | 12, A-366 | EC50 | > | 50 | uM | ALA5214731 | nM | Homo sapiens | |||
3. | (R)-PFI 2 hydrochloride | EUB0000196bCl | EC50 | > | 10 | uM | ALA5214705 | nM | Homo sapiens | |||
4. | OICR-9429 | 16d; OICR-9429 | % activity remaining | > | 90 | % | ALA5213720 | % | Homo sapiens | |||
5. | GSK343 | 6, GSK343 | IC50 | = | 240 | nM | ALA5214634 | 6.62 | nM | Homo sapiens | ||
6. | ALA3414619 | 21, UNC1999 | IC50 | = | 45 | nM | ALA5210592 | 7.35 | nM | Homo sapiens | ||
7. | ALA3414619 | 21, UNC1999 | IC50 | = | 124 | nM | ALA5210099 | 6.91 | nM | Homo sapiens | ||
8. | ALA5170450 | 8; MS8511 | INH | > | 50 | % | ALA5129691 | % | Homo sapiens | |||
9. | ALA3414574 | 20, EI1 | IC50 | = | 13 | nM | ALA5123969 | 7.89 | nM | Homo sapiens | ||
10. | ALA5197902 | OR-S0 | IC50 | = | 91 | nM | ALA5123963 | 7.04 | nM | Homo sapiens | ||
11. | ALA5185991 | 84 | IC50 | = | 7 | nM | ALA5123956 | 8.15 | nM | Homo sapiens | ||
12. | ALA5197386 | 79b; OR-S1 | IC50 | = | 0.47 | nM | ALA5123956 | 9.33 | nM | Homo sapiens | ||
13. | Valemetostat (DS-3201) | VALEMETOSTAT | IC50 | = | 0.44 | nM | ALA5123956 | 9.36 | nM | Homo sapiens | ||
14. | ALA5196227 | 32a; UNC1999 | IC50 | = | 45 | nM | ALA5123956 | 7.35 | nM | Homo sapiens | ||
15. | ALA5178720 | 20; ZLD-1122 | IC50 | = | 136.5 | nM | ALA5123952 | 6.87 | nM | Homo sapiens | ||
16. | ALA5203667 | 19b; ZLD-1039 | IC50 | = | 81 | nM | ALA5123946 | 7.09 | nM | Homo sapiens | ||
17. | ALA4637350 | SKLB1049 | IC50 | = | 84 | nM | ALA5123946 | 7.08 | nM | Homo sapiens | ||
18. | Ibiglustat | VENGLUSTAT | INH | = | 50 | % | ALA5119867 | % | Homo sapiens | |||
19. | Ibiglustat | VENGLUSTAT | INH | 0 | ALA5119830 | NA | % | Homo sapiens | ||||
20. | CPI-1205 | CPI-1205 | IC50 | = | 52 | nM | ALA4766109 | 7.28 | nM | Homo sapiens |