# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | astemizole | 52 (Astemizole) | Tm | = | 38.23 | degrees C | ALA3384851 | degrees C | Homo sapiens | |||
2. | astemizole | 52 (Astemizole) | Tm | = | 38.19 | degrees C | ALA3384850 | degrees C | Homo sapiens | |||
3. | astemizole | 52 (Astemizole) | Tm | = | 38.1 | degrees C | ALA3384849 | degrees C | Homo sapiens | |||
4. | astemizole | 52 (Astemizole) | Tm | = | 38.13 | degrees C | ALA3384848 | degrees C | Homo sapiens | |||
5. | astemizole | 52 (Astemizole) | Tm | = | 38.17 | degrees C | ALA3384847 | degrees C | Homo sapiens | |||
6. | astemizole | 52 (Astemizole) | Tm | = | 38.18 | degrees C | ALA3384846 | degrees C | Homo sapiens | |||
7. | astemizole | 52 (Astemizole) | Activity | 0 | ALA3384219 | Active | Homo sapiens | |||||
8. | astemizole | 52 (Astemizole) | Activity | 0 | ALA3384218 | Active | Homo sapiens | |||||
9. | astemizole | 52 (Astemizole) | Activity | 0 | ALA3384217 | Dose-dependent effect | Homo sapiens | |||||
10. | astemizole | 52 (Astemizole) | deltaTm | = | 1.64 | degrees C | ALA3382333 | degrees C | Homo sapiens | |||
11. | astemizole | 52 (Astemizole) | deltaTm | = | 2 | degrees C | ALA3382332 | degrees C | Homo sapiens | |||
12. | astemizole | 52 (Astemizole) | deltaTm | = | 3.44 | degrees C | ALA3382331 | degrees C | Homo sapiens | |||
13. | astemizole | 52 (Astemizole) | deltaTm | = | 4.29 | degrees C | ALA3382330 | degrees C | Homo sapiens | |||
14. | astemizole | 52 (Astemizole) | deltaTm | = | 4.08 | degrees C | ALA3382329 | degrees C | Homo sapiens | |||
15. | astemizole | 52 (Astemizole) | Ki | = | 23.01 | uM | ALA3382328 | 4.64 | nM | Homo sapiens | ||
16. | astemizole | 52 (Astemizole) | IC50 | = | 93.8 | uM | ALA3382328 | 4.03 | nM | Homo sapiens | ||
17. | ALA4850478 | 50 | pIC50 | = | 8.1 | ALA4834035 | 8.10 | nM | Homo sapiens | |||
18. | ALA4850478 | 50 | IC50 | = | 0.009 | uM | ALA4834035 | 8.05 | nM | Homo sapiens | ||
19. | ALA4847216 | 49 | pIC50 | = | 8.1 | ALA4834035 | 8.10 | nM | Homo sapiens | |||
20. | ALA4847216 | 49 | IC50 | = | 0.008 | uM | ALA4834035 | 8.10 | nM | Homo sapiens |