# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Wedelolactone | 1a | Kd | = | 2.82 | uM | ALA5237697 | 5.55 | nM | Homo sapiens | ||
2. | ALA5289498 | SAH-EZH2 | Kd | = | 0.32 | nM | ALA5237694 | 9.49 | nM | Homo sapiens | ||
3. | ALA4074159 | 1 | IC50 | = | 1.57 | uM | ALA5237690 | 5.80 | nM | Homo sapiens | ||
4. | ALA5273243 | EED666 | IC50 | = | 8.76 | uM | ALA5237690 | 5.06 | nM | Homo sapiens | ||
5. | ALA5269781 | 15; EED396, PDB 5H13 | IC50 | = | 11.58 | uM | ALA5237690 | 4.94 | nM | Homo sapiens | ||
6. | ALA4097892 | 1 | IC50 | = | 0.89 | uM | ALA5237690 | 6.05 | nM | Homo sapiens | ||
7. | ALA4096234 | 7 | IC50 | = | 0.32 | uM | ALA5237690 | 6.50 | nM | Homo sapiens | ||
8. | ALA5269445 | BR-001 | deltaTm | = | 6 | degrees C | ALA5237685 | degrees C | Homo sapiens | |||
9. | ALA5269445 | BR-001 | IC50 | = | 4.5 | nM | ALA5237684 | 8.35 | nM | Homo sapiens | ||
10. | A-395 | 2 | Kd | = | 1.5 | nM | ALA5237683 | 8.82 | nM | Homo sapiens | ||
11. | A-395 | 2 | deltaTm | = | 13 | degrees C | ALA5237682 | degrees C | Homo sapiens | |||
12. | ALA4755687 | 108 | pKd | = | 9.61 | ALA5231254 | 9.61 | nM | Homo sapiens | |||
13. | ALA5287008 | 6b | pKd | = | 9.02 | ALA5231254 | 9.02 | nM | Homo sapiens | |||
14. | ALA5275319 | 6a | pKd | = | 9.27 | ALA5231254 | 9.27 | nM | Homo sapiens | |||
15. | EED226 | 43 | IC50 | = | 45 | nM | ALA5231253 | 7.35 | nM | Homo sapiens | ||
16. | ALA4749741 | 109; UNC6852 | IC50 | = | 247 | nM | ALA5231252 | 6.61 | nM | Homo sapiens | ||
17. | ALA5288775 | H3K27me3 | Kd | = | 40 | uM | ALA5228444 | 4.40 | nM | Homo sapiens | ||
18. | ALA5287619 | JARID2-K116me3 | Kd | = | 3 | uM | ALA5228444 | 5.52 | nM | Homo sapiens | ||
19. | A-395 | 2 | deltaTm | = | 13 | degrees C | ALA5228435 | degrees C | Homo sapiens | |||
20. | ALA5268403 | 46; BR-001 | IC50 | = | 0.005 | uM | ALA5228433 | 8.35 | nM | Homo sapiens |