# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MLN2480 | SID174006384 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
2. | 6-piperidin-4-yloxy-2H-isoquinolin-1-one | 14C | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
3. | Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
4. | Sorafenib | 5 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
5. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
6. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
7. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
8. | ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
9. | CH5424802 | 18a, CH5424802 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
10. | Cediranib | 5, ZD-2171 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
11. | Tandutinib (MLN518) | 75 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
12. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
13. | CH4987655 | 24, CH4987655 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
14. | AZD1152 | 5 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
15. | Barasertib (AZD1152-HQPA) | 34 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
16. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
17. | ALA3991933 | Sapanisertib | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
18. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
19. | Foretinib (GSK1363089) | EXEL-2880/GSK-1363089 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens | ||
20. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991693 | Inactive | nM | Homo sapiens |