# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | conivaptan | Conivaptan | Ki | = | 44.4 | nM | ALA4201579 | 7.35 | nM | Rattus norvegicus | ||
2. | VNA932 | 2 | IC50 | = | 55 | nM | ALA4201594 | 7.26 | nM | Rattus norvegicus | ||
3. | ALA3272685 | 3 | Activity | = | 54 | % | ALA3284346 | % | Rattus norvegicus | |||
4. | ALA3272684 | 5 | Activity | = | 66 | % | ALA3284346 | % | Rattus norvegicus | |||
5. | ALA3272683 | 7 | Activity | = | 75 | % | ALA3284346 | % | Rattus norvegicus | |||
6. | ALA3245749 | [Leu4]oxytocin | Activity | = | 81 | % | ALA3284346 | % | Rattus norvegicus | |||
7. | [Phe³]OT | [Phe3]oxytocin | Activity | = | 90 | % | ALA3284346 | % | Rattus norvegicus | |||
8. | ALA3272685 | 3 | Activity | 0 | ALA3284339 | Not Determined | Rattus norvegicus | |||||
9. | ALA3272684 | 5 | Activity | = | 0.62 | U/mg | ALA3284339 | U/mg | Rattus norvegicus | |||
10. | ALA3272683 | 7 | Activity | = | 0.75 | U/mg | ALA3284339 | U/mg | Rattus norvegicus | |||
11. | ALA3245749 | [Leu4]oxytocin | Activity | = | 13 | U/mg | ALA3284339 | U/mg | Rattus norvegicus | |||
12. | [Phe³]OT | [Phe3]oxytocin | Activity | = | 39 | U/mg | ALA3284339 | U/mg | Rattus norvegicus | |||
13. | Oxytocin | Oxytocin | Activity | = | 533 | U/mg | ALA3285677 | U/mg | Rattus norvegicus | |||
14. | ALA3276119 | Deamino[carba-1]-oxytocin | Activity | = | 581 | U/mg | ALA3285677 | U/mg | Rattus norvegicus | |||
15. | ALA3276118 | [Carba-1]oxytocin | Activity | = | 177 | U/mg | ALA3285677 | U/mg | Rattus norvegicus | |||
16. | ALA3276115 | Hydroxy-oxytocin | Activity | = | 363 | U/mg | ALA3285677 | U/mg | Rattus norvegicus | |||
17. | ALA3276114 | Hydroxy[4-Thr]-oxytocin | Activity | = | 378 | U/mg | ALA3285677 | U/mg | Rattus norvegicus | |||
18. | ALA435716 | [Mpa1]oxytocin | Activity | = | 760 | U/mg | ALA3285676 | U/mg | Rattus norvegicus | |||
19. | Oxytocin | Oxytocin | Activity | = | 486 | U/mg | ALA3285676 | U/mg | Rattus norvegicus | |||
20. | ALA3276119 | Deamino[carba-1]-oxytocin | Activity | = | 921 | U/mg | ALA3285676 | U/mg | Rattus norvegicus |