# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2165443 | 39 | EC50 | = | 3400 | nM | ALA2168999 | 5.47 | nM | Homo sapiens | ||
2. | ALA2165444 | 43 | EC50 | = | 1200 | nM | ALA2168999 | 5.92 | nM | Homo sapiens | ||
3. | ALA2165445 | 44 | EC50 | > | 3000 | nM | ALA2168999 | nM | Homo sapiens | |||
4. | Nicotine | 2 | EC50 | = | 30000 | nM | ALA2168999 | 4.52 | nM | Homo sapiens | ||
5. | ALA1076903 | 9a table 2 | EC50 | = | 2200 | nM | ALA2168999 | 5.66 | nM | Homo sapiens | ||
6. | ALA2165443 | 39 | Efficacy | = | 120 | % | ALA2169197 | % | Homo sapiens | |||
7. | ALA2165444 | 43 | Efficacy | = | 120 | % | ALA2169197 | % | Homo sapiens | |||
8. | ALA2165445 | 44 | Efficacy | > | 80 | % | ALA2169197 | % | Homo sapiens | |||
9. | Nicotine | 2 | Efficacy | = | 90 | % | ALA2169197 | % | Homo sapiens | |||
10. | ALA1076903 | 9a table 2 | Efficacy | = | 110 | % | ALA2169197 | % | Homo sapiens | |||
11. | ALA2165443 | 39 | IC50 | > | 3000 | nM | ALA2169199 | nM | Homo sapiens | |||
12. | ALA2165444 | 43 | IC50 | > | 3000 | nM | ALA2169199 | nM | Homo sapiens | |||
13. | ALA2165445 | 44 | IC50 | > | 3000 | nM | ALA2169199 | nM | Homo sapiens | |||
14. | Nicotine | 2 | IC50 | 0 | ALA2169199 | Not Determined | Homo sapiens | |||||
15. | ALA1076903 | 9a table 2 | IC50 | 0 | ALA2169199 | Not Determined | Homo sapiens | |||||
16. | ALA2165443 | 39 | Efficacy | > | 70 | % | ALA2169201 | % | Homo sapiens | |||
17. | ALA2165444 | 43 | Efficacy | > | 70 | % | ALA2169201 | % | Homo sapiens | |||
18. | ALA2165445 | 44 | Efficacy | > | 30 | % | ALA2169201 | % | Homo sapiens | |||
19. | Nicotine | 2 | Efficacy | 0 | ALA2169201 | Not Determined | Homo sapiens | |||||
20. | ALA1076903 | 9a table 2 | Efficacy | 0 | ALA2169201 | Not Determined | Homo sapiens |