| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2031263 | 56 | Activity | 0 | ALA4274805 | Not Active | Renilla reniformis | |||||
| 2. |  ALA4287905 | MRT-92 | Activity | 0 | ALA4274805 | Not Active | Renilla reniformis | |||||
| 3. |  MRT-83 hydrochloride | 4; ST8117 | Activity | 0 | ALA4274805 | Not Active | Renilla reniformis | |||||
| 4. |  ALA4283244 | 3; ST8115 | Activity | 0 | ALA4274805 | Not Active | Renilla reniformis | |||||
| 5. |  Vismodegib (GDC-0449) | 101, GDC-0449 | Activity | 0 | ALA4274805 | Not Active | Renilla reniformis | |||||
| 6. |  ALA1221983 | 2, SAG | Activity | < | 20 | % | ALA3860358 | % | Renilla reniformis | |||
| 7. |  GSA-10 | 1; GSA-10 | Activity | < | 20 | % | ALA3860358 | % | Renilla reniformis | |||
| 8. |  ALA3927217 | 20 | Activity | < | 20 | % | ALA3860358 | % | Renilla reniformis | |||
| 9. |  ALA3971451 | 25 | Activity | < | 20 | % | ALA3860358 | % | Renilla reniformis | |||
| 10. |  ALA1909414 | SB-590885-AAD | AC50 | = | 29.063 | uM | ALA2303648 | 4.54 | Phenotype: Inhibitor; Curve_Description: Partial curve; partial efficacy | nM | Renilla reniformis | |
| 11. |  ALA1909376 | SB-759335-B | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Activator; Curve_Description: None | nM | Renilla reniformis | ||
| 12. |  ALA506153 | 2 | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Inactive; Curve_Description: None | nM | Renilla reniformis | ||
| 13. |  ALA273564 | 8d | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Inactive; Curve_Description: None | nM | Renilla reniformis | ||
| 14. |  ALA456252 | 27 | AC50 | = | 46.062 | uM | ALA2303648 | 4.34 | Phenotype: Inhibitor; Curve_Description: Partial curve; partial efficacy; poor fit | nM | Renilla reniformis | |
| 15. |  ALA458415 | 33 | AC50 | = | 23.085 | uM | ALA2303648 | 4.64 | Phenotype: Inhibitor; Curve_Description: Partial curve; partial efficacy; poor fit | nM | Renilla reniformis | |
| 16. |  ALA467581 | 13 | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Inactive; Curve_Description: None | nM | Renilla reniformis | ||
| 17. |  ALA205966 | 8d | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Inactive; Curve_Description: None | nM | Renilla reniformis | ||
| 18. |  ALA511765 | 11 | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Inactive; Curve_Description: None | nM | Renilla reniformis | ||
| 19. |  ALA1794069 | 22 | AC50 | = | 20.575 | uM | ALA2303648 | 4.69 | Phenotype: Inhibitor; Curve_Description: Partial curve; partial efficacy | nM | Renilla reniformis | |
| 20. |  3-[(2-{[1-(N,N-Dimethylglycyl)-6-Methoxy-4,4-Dimethyl-1,2,3,4-Tetrahydroquinolin-7-Yl]amino}-7h-Pyrrolo[2,3-D]pyrimidin-4-Yl)amino]thiophene-2-Carboxamide | 28 | AC50 | = | 0 | uM | ALA2303648 | Phenotype: Inactive; Curve_Description: None | nM | Renilla reniformis |
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