# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3617067 | HNTX-IV | IC50 | = | 375 | nM | ALA3618947 | 6.43 | nM | Rattus norvegicus | ||
2. | ALA3589861 | (R)-9 | INH | 0 | ALA3592078 | Not Active | % | Rattus norvegicus | ||||
3. | ALA3589861 | (R)-9 | V1/2 | = | -72.84 | mV | ALA3592074 | mV | Rattus norvegicus | |||
4. | ALA3589861 | (R)-9 | V1/2 | = | -32.48 | mV | ALA3592070 | mV | Rattus norvegicus | |||
5. | ALA3589861 | (R)-9 | INH | 0 | ALA3592066 | Active | % | Rattus norvegicus | ||||
6. | Tetrodotoxin | TETRODOTOXIN | IC50 | = | 15 | nM | ALA3880174 | 7.82 | nM | Rattus norvegicus | ||
7. | Lacosamide | (R)18 | IC50 | = | 415 | nM | ALA4257756 | 6.38 | nM | Rattus norvegicus | ||
8. | ICA 121431 | 16, ICA-121431 | IC50 | = | 6 | nM | ALA4257699 | 8.22 | nM | Rattus norvegicus | ||
9. | ALA5190671 | Hact-2 | Activity | 0 | ALA5125243 | NA | Rattus norvegicus | |||||
10. | ALA5084333 | alpha 7 | EC50 | = | 170.2 | nM | ALA5037532 | 6.77 | nM | Rattus norvegicus | ||
11. | ALA5082582 | alpha6 | EC50 | = | 105.6 | nM | ALA5037532 | 6.98 | nM | Rattus norvegicus | ||
12. | ALA5093878 | alpha 5 | EC50 | = | 9.4 | nM | ALA5037532 | 8.03 | nM | Rattus norvegicus | ||
13. | ALA5077579 | alpha 4 | EC50 | = | 12.9 | nM | ALA5037532 | 7.89 | nM | Rattus norvegicus | ||
14. | ALA5091623 | alpha 3 | EC50 | = | 138.9 | nM | ALA5037532 | 6.86 | nM | Rattus norvegicus | ||
15. | ALA5083412 | alpha 2 | EC50 | = | 127.7 | nM | ALA5037532 | 6.89 | nM | Rattus norvegicus | ||
16. | ALA5091679 | alpha 1 | EC50 | = | 135.4 | nM | ALA5037532 | 6.87 | nM | Rattus norvegicus | ||
17. | Lacosamide | (R)18 | IC50 | = | 415 | nM | ALA2328118 | 6.38 | nM | Rattus norvegicus | ||
18. | ALA2324353 | 31 | IC50 | < | 2 | uM | ALA2328108 | nM | Rattus norvegicus | |||
19. | ALA1917113 | 6, D9K13 | INH | = | 29.1 | % | ALA1918335 | % | Rattus norvegicus | |||
20. | ALA1917257 | 8, D9K13 linear | INH | 0 | ALA1918438 | Not Active | % | Rattus norvegicus |