# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4460144 | JBP923 | Ki | = | 2.5 | mM | ALA4375725 | nM | Homo sapiens | |||
2. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Ki | = | 36 | mM | ALA4375725 | nM | Homo sapiens | |||
3. | ALA4460144 | JBP923 | IC50 | = | 1.76 | mM | ALA4375703 | nM | Homo sapiens | |||
4. | ALA4540326 | 12a; J3V | IC50 | = | 2.9 | mM | ALA4375703 | nM | Homo sapiens | |||
5. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | IC50 | = | 18.2 | mM | ALA4375703 | nM | Homo sapiens | |||
6. | ALA4460144 | JBP923 | Km | = | 0.65 | mM | ALA4375702 | nM | Homo sapiens | |||
7. | ALA4540326 | 12a; J3V | Km | = | 0.86 | mM | ALA4375702 | nM | Homo sapiens | |||
8. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Km | = | 2.53 | mM | ALA4375702 | nM | Homo sapiens | |||
9. | ALA4460144 | JBP923 | Drug uptake | 0 | ALA4375695 | Not Active | Homo sapiens | |||||
10. | ALA4540326 | 12a; J3V | Drug uptake | 0 | ALA4375695 | Not Active | Homo sapiens | |||||
11. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Drug uptake | 0 | ALA4375695 | Not Active | Homo sapiens | |||||
12. | ALA4460144 | JBP923 | Drug uptake | 0 | ALA4375694 | Not Active | Homo sapiens | |||||
13. | ALA4540326 | 12a; J3V | Drug uptake | 0 | ALA4375694 | Not Active | Homo sapiens | |||||
14. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Drug uptake | 0 | ALA4375694 | Not Active | Homo sapiens | |||||
15. | ALA4460144 | JBP923 | Drug uptake | 0 | ALA4375693 | Active | Homo sapiens | |||||
16. | ALA4540326 | 12a; J3V | Drug uptake | 0 | ALA4375693 | Active | Homo sapiens | |||||
17. | ALA2229108 | 28, cyclo-(Ser-trans-4-OH-Pro) | Drug uptake | 0 | ALA4375693 | Active | Homo sapiens | |||||
18. | ALA4168781 | 11 | Ratio | 0 | ALA4156375 | Not Determined | Homo sapiens | |||||
19. | ALA4173276 | 10 | Ratio | 0 | ALA4156375 | Not Determined | Homo sapiens | |||||
20. | ALA4165361 | 9 | Ratio | 0 | ALA4156375 | Not Determined | Homo sapiens |