| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3527165 | LK, LK-980 | Activity | = | 10.1 | ug | ALA3539028 | ug | Homo sapiens | |||
| 2. |  IRAK3 PROTAC 23 | 23 | INH | < | 40 | % | ALA4729480 | % | Homo sapiens | |||
| 3. |  PF-04691502 | 3 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 4. |  6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 5. |  RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 6. |  Pelitinib | EKB-569 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 7. |  CH4987655 | 24, CH4987655 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 8. |  AZD2014 | 21, AZD2014 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 9. |  Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 10. |  Danusertib (PHA-739358) | 9d | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 11. |  Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 12. |  ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 13. |  OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 14. |  Savolitinib (AZD6094) | 28 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 15. |  Sorafenib | 5 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 16. |  Tandutinib (MLN518) | 75 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 17. |  Linifanib (ABT-869) | 17p, ABT-869 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 18. |  Afuresertib (GSK2110183) | AFURESERTIB | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 19. |  avutometinib | 1, CH5126766/RO5126766 | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens | ||
| 20. |  ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991691 | Inactive | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!