# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -0.5 | degrees C | ALA5236408 | degrees C | Homo sapiens | |||
2. | ALA5267793 | 9d | deltaTm | = | 0 | degrees C | ALA5236408 | degrees C | Homo sapiens | |||
3. | ALA4746865 | 23 | IC50 | = | 370 | nM | ALA5231297 | 6.43 | nM | Homo sapiens | ||
4. | ALA5278697 | 24a; ACB11 | IC50 | = | 770 | nM | ALA5231297 | 6.11 | nM | Homo sapiens | ||
5. | PFI-3 | 72; PFI-3 | dTm | = | 9.2 | K | ALA5214138 | K | Homo sapiens | |||
6. | PFI-3 | 72; PFI-3 | Kd | = | 89 | nM | ALA5210533 | 7.05 | nM | Homo sapiens | ||
7. | PFI-3 | 72; PFI-3 | EC50 | < | 1000 | nM | ALA5210237 | nM | Homo sapiens | |||
8. | ALA5204783 | 8m | deltaTm | = | 1 | degrees C | ALA5162543 | degrees C | Homo sapiens | |||
9. | ALA5206088 | 8l; XY153 | deltaTm | = | 1 | degrees C | ALA5162543 | degrees C | Homo sapiens | |||
10. | ALA5205742 | 8k | deltaTm | = | 0.75 | degrees C | ALA5162543 | degrees C | Homo sapiens | |||
11. | ALA5178480 | 8j | deltaTm | = | -0.25 | degrees C | ALA5162543 | degrees C | Homo sapiens | |||
12. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 0.25 | degrees C | ALA5162543 | degrees C | Homo sapiens | |||
13. | ALA5204783 | 8m | deltaTm | = | 1 | degrees C | ALA5162542 | degrees C | Homo sapiens | |||
14. | ALA5206088 | 8l; XY153 | deltaTm | = | 1 | degrees C | ALA5162542 | degrees C | Homo sapiens | |||
15. | ALA5205742 | 8k | deltaTm | = | 0.5 | degrees C | ALA5162542 | degrees C | Homo sapiens | |||
16. | ALA5178480 | 8j | deltaTm | = | 0.75 | degrees C | ALA5162542 | degrees C | Homo sapiens | |||
17. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -0.25 | degrees C | ALA5162542 | degrees C | Homo sapiens | |||
18. | ALA5179520 | 9g; Y08284 | deltaTm | = | -0.5 | degrees C | ALA5156584 | degrees C | Homo sapiens | |||
19. | ALA5204688 | 9d | deltaTm | = | -0.3 | degrees C | ALA5156584 | degrees C | Homo sapiens | |||
20. | ALA5192803 | 9c | deltaTm | = | -0.3 | degrees C | ALA5156584 | degrees C | Homo sapiens |