# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4284872 | 19 | Emax | = | 89 | % | ALA4252017 | % | Homo sapiens | |||
2. | ALA4083687 | 3 | Emax | = | 108 | % | ALA4252017 | % | Homo sapiens | |||
3. | ALA4284872 | 19 | EC50 | = | 0.6 | uM | ALA4252017 | 6.22 | nM | Homo sapiens | ||
4. | ALA4083687 | 3 | EC50 | = | 0.3 | uM | ALA4252017 | 6.52 | nM | Homo sapiens | ||
5. | ALA4074873 | 20-AM-1488 | Emax | = | 104.3 | % | ALA4219935 | % | Homo sapiens | |||
6. | ALA4074873 | 20-AM-1488 | EC50 | = | 0.171 | uM | ALA4219929 | 6.77 | nM | Homo sapiens | ||
7. | ALA4070615 | 32; AM-3607 | EC50 | = | 16 | nM | ALA4219620 | 7.80 | nM | Homo sapiens | ||
8. | ALA4074873 | 20-AM-1488 | EC50 | = | 171 | nM | ALA4219620 | 6.77 | nM | Homo sapiens | ||
9. | Gelsemine | gelsemine | IC50 | = | 30 | uM | ALA4219611 | 4.52 | nM | Homo sapiens | ||
10. | ALA4103909 | 6i | IC50 | = | 0.043 | uM | ALA3998490 | 7.37 | nM | Homo sapiens | ||
11. | ALA4079657 | 6h | IC50 | = | 0.046 | uM | ALA3998490 | 7.34 | nM | Homo sapiens | ||
12. | ALA4068867 | 6b | IC50 | = | 0.116 | uM | ALA3998490 | 6.94 | nM | Homo sapiens | ||
13. | ALA4102677 | 6a | IC50 | = | 0.056 | uM | ALA3998490 | 7.25 | nM | Homo sapiens | ||
14. | ALA4069635 | 4 | IC50 | = | 6.53 | uM | ALA3998490 | 5.18 | nM | Homo sapiens | ||
15. | ALA4096857 | 3 | IC50 | = | 0.311 | uM | ALA3998490 | 6.51 | nM | Homo sapiens | ||
16. | ALA4060962 | 2 | IC50 | = | 0.097 | uM | ALA3998490 | 7.01 | nM | Homo sapiens | ||
17. | ALA4089150 | 1 | IC50 | = | 0.08 | uM | ALA3998490 | 7.10 | nM | Homo sapiens | ||
18. | [³H]strychnine | Strychnine | IC50 | = | 0.058 | uM | ALA3998490 | 7.24 | nM | Homo sapiens | ||
19. | ALA4061219 | 6k | pIC50 | = | 5.83 | ALA3998488 | 5.83 | nM | Homo sapiens | |||
20. | ALA4096505 | 6j | pIC50 | = | 6.18 | ALA3998488 | 6.18 | nM | Homo sapiens |