# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | N,N,2-Trimethyl-5-nitrobenzenesulfonamide | BRL-50481 | IC50 | = | 62 | uM | ALA5227540 | 4.21 | nM | Homo sapiens | ||
2. | ALA4129844 | (R)-3 | IC50 | = | 0.596 | uM | ALA5226665 | 6.22 | nM | Homo sapiens | ||
3. | ALA4128481 | (S)-3 | IC50 | = | 0.009 | uM | ALA5226665 | 8.05 | nM | Homo sapiens | ||
4. | ALA3601546 | 2 | IC50 | = | 0.13 | uM | ALA5226628 | 6.89 | nM | Homo sapiens | ||
5. | ALA5269084 | 14 | IC50 | = | 0.219 | uM | ALA5226628 | 6.66 | nM | Homo sapiens | ||
6. | ALA5180169 | 2g | IC50 | = | 354 | nM | ALA5168612 | 6.45 | nM | Homo sapiens | ||
7. | ALA5171560 | 33a | IC50 | > | 10000 | nM | ALA5159512 | nM | Homo sapiens | |||
8. | ALA4471352 | 4e | IC50 | > | 10000 | nM | ALA4404709 | nM | Homo sapiens | |||
9. | BPN14770 | ZATOLMILAST | INH | 0 | ALA4397278 | Not Active | % | Homo sapiens | ||||
10. | BAY-60-7550 | table 2 BAY-607550 | INH | = | 86 | % | ALA4395200 | % | Homo sapiens | |||
11. | BAY-60-7550 | table 2 BAY-607550 | INH | = | 55 | % | ALA4395178 | % | Homo sapiens | |||
12. | BAY-60-7550 | table 2 BAY-607550 | INH | = | 16 | % | ALA4395156 | % | Homo sapiens | |||
13. | ALA4468513 | 3b; DRILS-1765 | INH | = | 23 | % | ALA4395100 | % | Homo sapiens | |||
14. | ALA1513993 | 1, BAY-736691 | IC50 | = | 50 | nM | ALA4385789 | 7.30 | nM | Homo sapiens | ||
15. | ALA4436823 | 1k | IC50 | = | 2 | uM | ALA4385789 | 5.70 | nM | Homo sapiens | ||
16. | ALA4564974 | 1j | IC50 | = | 1.2 | uM | ALA4385789 | 5.92 | nM | Homo sapiens | ||
17. | ALA4457086 | 1i | IC50 | = | 0.7 | uM | ALA4385789 | 6.16 | nM | Homo sapiens | ||
18. | ALA4435082 | 1h | IC50 | = | 2.4 | uM | ALA4385789 | 5.62 | nM | Homo sapiens | ||
19. | ALA4445082 | 1g | IC50 | = | 7.8 | uM | ALA4385789 | 5.11 | nM | Homo sapiens | ||
20. | ALA4515145 | 1f | IC50 | = | 10 | uM | ALA4385789 | 5.00 | nM | Homo sapiens |