# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288161 | [18F]BIT1 | IC50 | = | 3.3 | nM | ALA5227558 | 8.48 | nM | Homo sapiens | ||
2. | ALA5284717 | [18F]TA5 | IC50 | = | 3 | nM | ALA5227558 | 8.52 | nM | Homo sapiens | ||
3. | ALA5272525 | [18F]TA4 | IC50 | = | 913 | nM | ALA5227558 | 6.04 | nM | Homo sapiens | ||
4. | ALA5286170 | [18F]TA3 | IC50 | = | 11.4 | nM | ALA5227558 | 7.94 | nM | Homo sapiens | ||
5. | ALA3092563 | 19, [18F]-19 | IC50 | = | 1.4 | nM | ALA5227558 | 8.85 | nM | Homo sapiens | ||
6. | PF-05085727 | 1 | IC50 | = | 2.3 | nM | ALA5227557 | 8.64 | nM | Homo sapiens | ||
7. | PF 05180999 | 15, PF-999 | IC50 | = | 1 | nM | ALA5227557 | 9.00 | nM | Homo sapiens | ||
8. | ALA3092565 | 2, ND-7001 | IC50 | = | 1 | nM | ALA5227557 | 9.00 | nM | Homo sapiens | ||
9. | N,N,2-Trimethyl-5-nitrobenzenesulfonamide | BRL-50481 | IC50 | = | 62 | uM | ALA5227542 | 4.21 | nM | Homo sapiens | ||
10. | ALA5268162 | 53 | IC50 | = | 0.001 | uM | ALA5226640 | 9.29 | nM | Homo sapiens | ||
11. | ALA5274203 | 52 | IC50 | = | 0.005 | uM | ALA5226640 | 8.29 | nM | Homo sapiens | ||
12. | ALA4087340 | 5 | IC50 | = | 0.48 | uM | ALA5226640 | 6.32 | nM | Homo sapiens | ||
13. | ALA4068452 | 23 | IC50 | = | 0.024 | uM | ALA5226640 | 7.62 | nM | Homo sapiens | ||
14. | ALA5276846 | 42 | IC50 | = | 0.003 | uM | ALA5226637 | 8.48 | nM | Homo sapiens | ||
15. | ALA5267226 | 41 | IC50 | = | 0.003 | uM | ALA5226637 | 8.52 | nM | Homo sapiens | ||
16. | ALA5269828 | 40 | IC50 | = | 0.005 | uM | ALA5226637 | 8.35 | nM | Homo sapiens | ||
17. | ALA5268661 | 24; Bay-60-7550 | IC50 | = | 0.005 | uM | ALA5226636 | 8.33 | nM | Homo sapiens | ||
18. | BAY-299 | 5b; atropisomer 2 | % of control | = | 49 | % | ALA5214109 | % | Homo sapiens | |||
19. | TP-472 | 1; TP-472 | % of control | = | 25 | % | ALA5214184 | % | Homo sapiens | |||
20. | ALA4518342 | EUB0000744 | Ki | > | 100 | uM | ALA5213972 | nM | Homo sapiens |