| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  GSK2334470 | (3S,6R)-28d, GSK-2334470 | IC50 | = | 2.5 | nM | ALA5210316 | 8.60 | nM | Homo sapiens | ||
| 2. | GSK2334470 | (3S,6R)-28d, GSK-2334470 | IC50 | = | 113 | nM | ALA5209904 | 6.95 | nM | Homo sapiens | ||
| 3. |  BX-795 | BX-795 | IC50 | = | 6 | nM | ALA5131709 | 8.22 | nM | Homo sapiens | ||
| 4. |  ALA4564126 | 18 | INH | <= | 16 | % | ALA4427670 | % | Homo sapiens | |||
| 5. | ALA4564126 | 18 | IC50 | >= | 5 | uM | ALA4427726 | nM | Homo sapiens | |||
| 6. |  JTE-952 | JTE-952; (S)-8b | IC50 | > | 1000 | nM | ALA4424900 | nM | Homo sapiens | |||
| 7. |  ALA1422005 | SID26729800 | Activity | 0 | ALA4419260 | Not Active | Homo sapiens | |||||
| 8. |  ALA4588492 | 120; Fig 3 Cpd 4 | Activity | 0 | ALA4419260 | Not Active | Homo sapiens | |||||
| 9. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405507 | % | Homo sapiens | |||
| 10. |  AZD7648 | Example 16; AZD7648 | IC50 | > | 8.3 | uM | ALA4403985 | nM | Homo sapiens | |||
| 11. |  ALA4592040 | Ref 18, RS1 | Kd | = | 1.5 | uM | ALA4402906 | 5.82 | nM | Homo sapiens | ||
| 12. |  ALA4536012 | 20c | INH | = | -5.07 | % | ALA4395902 | % | Homo sapiens | |||
| 13. |  ALA4559936 | (+/-)-6 | Activity | = | 41 | % | ALA4391497 | % | Homo sapiens | |||
| 14. |  ALA4564973 | 50 | INH | = | 34 | % | ALA4389871 | % | Homo sapiens | |||
| 15. |  ALA4555459 | 43 | INH | = | 41 | % | ALA4389394 | % | Homo sapiens | |||
| 16. |  ALA4545456 | 24 | INH | = | 8.5 | % | ALA4387320 | % | Homo sapiens | |||
| 17. |  Abemaciclib | ABEMACICLIB | INH | = | 1 | % | ALA4387320 | % | Homo sapiens | |||
| 18. |  ALA4473365 | 7c | Activity | = | 94 | % | ALA4382675 | % | Homo sapiens | |||
| 19. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379288 | nM | Homo sapiens | |||
| 20. |  ALA2348350 | 15u | Activity | = | 96 | % | ALA4806684 | % | Homo sapiens |
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