# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 4-[[[2-[(4-fluorophenyl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carbonyl]amino]methyl]benzoic acid | 47 | IC50 | = | 24.3 | nM | ALA5168388 | 7.61 | nM | Mus musculus | ||
2. | ALA5208220 | 35 | IC50 | = | 336.2 | nM | ALA5168388 | 6.47 | nM | Mus musculus | ||
3. | ALA5188328 | 27 | IC50 | = | 66.7 | nM | ALA5168388 | 7.18 | nM | Mus musculus | ||
4. | E7046 (ER-886406) | BDBM119448 | IC50 | = | 101.2 | nM | ALA5168388 | 7.00 | nM | Mus musculus | ||
5. | ALA5195058 | 22 | IC50 | = | 50.1 | nM | ALA5168388 | 7.30 | nM | Mus musculus | ||
6. | ALA5179032 | 18 | IC50 | = | 29 | nM | ALA5168388 | 7.54 | nM | Mus musculus | ||
7. | ALA5181722 | 17 | IC50 | = | 19.8 | nM | ALA5168388 | 7.70 | nM | Mus musculus | ||
8. | ALA5189703 | 36 | IC50 | = | 2.8 | nM | ALA5168388 | 8.55 | nM | Mus musculus | ||
9. | ALA5205440 | 39 | IC50 | 0 | ALA5168388 | ND | Mus musculus | |||||
10. | ALA5179874 | 41 | IC50 | 0 | ALA5168388 | ND | Mus musculus | |||||
11. | Grapiprant (CJ-023,423) | GRAPIPRANT | pA2 | = | 8.11 | ALA3997101 | 8.11 | nM | Mus musculus | |||
12. | ALA4099851 | 4j; AAT-008 | pA2 | = | 9 | ALA3997101 | 9.00 | nM | Mus musculus | |||
13. | ALA4550862 | 65 | IC50 | = | 219.7 | nM | ALA4380430 | 6.66 | nM | Mus musculus | ||
14. | ALA4455965 | 64 | IC50 | = | 130 | nM | ALA4380430 | 6.89 | nM | Mus musculus | ||
15. | ALA4576681 | 62 | IC50 | = | 33.7 | nM | ALA4380430 | 7.47 | nM | Mus musculus | ||
16. | ALA4591792 | 61 | IC50 | = | 70.9 | nM | ALA4380430 | 7.15 | nM | Mus musculus | ||
17. | EP4 receptor antagonist 1 | 59 | IC50 | = | 16.2 | nM | ALA4380430 | 7.79 | nM | Mus musculus | ||
18. | ALA4548291 | 58 | IC50 | = | 42.1 | nM | ALA4380430 | 7.38 | nM | Mus musculus | ||
19. | ALA4440382 | 57 | IC50 | = | 57.6 | nM | ALA4380430 | 7.24 | nM | Mus musculus | ||
20. | ALA4564092 | 56 | IC50 | = | 27.5 | nM | ALA4380430 | 7.56 | nM | Mus musculus |