# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3291291 | 4 | IC50 | = | 5.7 | uM | ALA3295791 | 5.24 | nM | Homo sapiens | ||
2. | ALA3291290 | 3 | IC50 | = | 2.3 | uM | ALA3295791 | 5.64 | nM | Homo sapiens | ||
3. | ALA3237861 | 2 | IC50 | = | 29 | nM | ALA3295791 | 7.54 | nM | Homo sapiens | ||
4. | ALA3237860 | 1 | IC50 | = | 5.7 | nM | ALA3295791 | 8.24 | nM | Homo sapiens | ||
5. | ALA491636 | 1 | IC50 | = | 1440 | nM | ALA3295791 | 5.84 | nM | Homo sapiens | ||
6. | Carfilzomib | 2 | IC50 | = | 8.6 | nM | ALA3266057 | 8.07 | nM | Homo sapiens | ||
7. | Bortezomib (PS-341) | 15 | IC50 | = | 7.14 | nM | ALA3266057 | 8.15 | nM | Homo sapiens | ||
8. | ALA3262768 | 22h | IC50 | 0 | ALA3266057 | Not Determined | Homo sapiens | |||||
9. | ALA3262767 | 22f | IC50 | 0 | ALA3266057 | Not Determined | Homo sapiens | |||||
10. | ALA3262766 | 20h | IC50 | = | 0.11 | uM | ALA3266057 | 6.96 | nM | Homo sapiens | ||
11. | ALA3262765 | 20f | IC50 | = | 0.17 | uM | ALA3266057 | 6.77 | nM | Homo sapiens | ||
12. | ALA3262764 | 18n | IC50 | 0 | ALA3266057 | Not Determined | Homo sapiens | |||||
13. | ALA3262763 | 18m | IC50 | 0 | ALA3266057 | Not Determined | Homo sapiens | |||||
14. | ALA3262762 | 18l | IC50 | = | 0.63 | uM | ALA3266057 | 6.20 | nM | Homo sapiens | ||
15. | ALA3262761 | 18k | IC50 | = | 0.95 | uM | ALA3266057 | 6.02 | nM | Homo sapiens | ||
16. | ALA3262760 | 18j | IC50 | 0 | ALA3266057 | Not Determined | Homo sapiens | |||||
17. | ALA3262759 | 18i | IC50 | 0 | ALA3266057 | Not Determined | Homo sapiens | |||||
18. | ALA3262758 | 18h | IC50 | = | 0.19 | uM | ALA3266057 | 6.72 | nM | Homo sapiens | ||
19. | ALA3262757 | 18g | IC50 | = | 0.36 | uM | ALA3266057 | 6.44 | nM | Homo sapiens | ||
20. | ALA3262756 | 18f | IC50 | = | 0.22 | uM | ALA3266057 | 6.66 | nM | Homo sapiens |