# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Busulfan | Busulfan | Activity | 0 | ALA3295785 | Not Active | Homo sapiens | |||||
2. | ALA3291023 | mBBG | Activity | 0 | ALA3295785 | Active | Homo sapiens | |||||
3. | ALA3291022 | pBBG | Activity | 0 | ALA3295785 | Active | Homo sapiens | |||||
4. | m-Iodobenzylguanidine hemisulfate salt | 2b | Activity | = | 98 | % | ALA3295785 | % | Homo sapiens | |||
5. | Busulfan | Busulfan | Activity | 0 | ALA3295782 | Active | Homo sapiens | |||||
6. | m-Iodobenzylguanidine hemisulfate salt | 2b | Activity | 0 | ALA3295782 | Active | Homo sapiens | |||||
7. | ALA3291023 | mBBG | Activity | 0 | ALA3293098 | Dose-dependent effect | Homo sapiens | |||||
8. | ALA3291022 | pBBG | Activity | 0 | ALA3293098 | Dose-dependent effect | Homo sapiens | |||||
9. | Rucaparib | 63, AG-014699 | IC50 | = | 59.709 | uM | ALA2363637 | 4.22 | nM | Homo sapiens | ||
10. | CCT 018159 | 3a CCT018159 | IC50 | = | 63.723 | uM | ALA2363637 | 4.20 | nM | Homo sapiens | ||
11. | TW-37 | 5, TW-37 | IC50 | = | 0.664 | uM | ALA2363637 | 6.18 | nM | Homo sapiens | ||
12. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 10.224 | uM | ALA2363637 | 4.99 | nM | Homo sapiens | ||
13. | PF-4708671 | SID137275978 | IC50 | = | 612.802 | uM | ALA2363637 | nM | Homo sapiens | |||
14. | Avagacestat | 80 BMS-708163 | IC50 | = | 25.605 | uM | ALA2363637 | 4.59 | nM | Homo sapiens | ||
15. | EHT 1864 | SID137275837 | IC50 | = | 52.935 | uM | ALA2363637 | 4.28 | nM | Homo sapiens | ||
16. | CCT007093 | A17 | IC50 | = | 116.643 | uM | ALA2363637 | nM | Homo sapiens | |||
17. | AZD6482 | AZD-6482 | IC50 | = | 79.088 | uM | ALA2363637 | 4.10 | nM | Homo sapiens | ||
18. | ALA191384 | figure 1, 6 | IC50 | = | 10.87 | uM | ALA2363637 | 4.96 | nM | Homo sapiens | ||
19. | ALA289228 | 1, R-115777 | IC50 | = | 29.644 | uM | ALA2363637 | 4.53 | nM | Homo sapiens | ||
20. | Epothilone B | Epothilone B | IC50 | = | 0.019 | uM | ALA2363637 | 7.72 | nM | Homo sapiens |