# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Imatinib Mesylate (STI571) | 1, Gleevec | IC50 | = | 100 | nM | ALA5253983 | 7.00 | nM | Homo sapiens | ||
2. | ALA4527555 | 1 | IC50 | < | 10 | nM | ALA5253982 | nM | Homo sapiens | |||
3. | Imatinib Mesylate (STI571) | 1, Gleevec | IC50 | = | 100 | nM | ALA5253981 | 7.00 | nM | Homo sapiens | ||
4. | ALA2313790 | 18 | IC50 | = | 28 | nM | ALA5253975 | 7.55 | nM | Homo sapiens | ||
5. | ALA3318100 | 22 | IC50 | = | 28 | nM | ALA5253975 | 7.55 | nM | Homo sapiens | ||
6. | ALA4527555 | 1 | IC50 | = | 14 | nM | ALA5253975 | 7.85 | nM | Homo sapiens | ||
7. | ALA4527555 | 1 | INH | = | 50 | % | ALA5253951 | % | Homo sapiens | |||
8. | ALA1614701 | AZD-6244 | IC50 | = | 0.456 | uM | ALA2363366 | 6.34 | nM | Homo sapiens | ||
9. | SB590885 | 33, SB-590885 | IC50 | = | 43.842 | uM | ALA2363366 | 4.36 | nM | Homo sapiens | ||
10. | PD0325901 | 34, PD-0325901 | IC50 | = | 0.095 | uM | ALA2363366 | 7.02 | nM | Homo sapiens | ||
11. | AZD8055 | 10, AZD-8055 | IC50 | = | 0.18 | uM | ALA2363366 | 6.74 | nM | Homo sapiens | ||
12. | GDC-0941 | 17, GDC-0941 | IC50 | = | 2.027 | uM | ALA2363366 | 5.69 | nM | Homo sapiens | ||
13. | BEZ235 | SID124898663 | IC50 | = | 0.036 | uM | ALA2363366 | 7.45 | nM | Homo sapiens | ||
14. | Palbociclib | 43(table 3) | IC50 | = | 0.258 | uM | ALA2363366 | 6.59 | nM | Homo sapiens | ||
15. | MK-2206 | 17 | IC50 | = | 4.142 | uM | ALA2363366 | 5.38 | nM | Homo sapiens | ||
16. | Ro 3306 | 28 | IC50 | = | 111.089 | uM | ALA2363366 | nM | Homo sapiens | |||
17. | ZM-447439 | 2 | IC50 | = | 1.755 | uM | ALA2363366 | 5.76 | nM | Homo sapiens | ||
18. | PD173074 | 12 | IC50 | = | 4.533 | uM | ALA2363366 | 5.34 | nM | Homo sapiens | ||
19. | Nutlin-3a | Nutlin-3 | IC50 | = | 34.607 | uM | ALA2363366 | 4.46 | nM | Homo sapiens | ||
20. | Wee1 inhibitor | 23 | IC50 | = | 8.773 | uM | ALA2363366 | 5.06 | nM | Homo sapiens |