# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3086474 | 1, Cis diastereomer | Ratio EC50 | = | 8 | ALA3089288 | Homo sapiens | |||||
2. | ALA3086474 | 1, Cis diastereomer | FC | = | 45 | ALA3089289 | Homo sapiens | |||||
3. | ALA3086473 | 1a, GAT106 | Activity | 0 | ALA3089296 | Not Active | Homo sapiens | |||||
4. | ALA3086472 | 1b, GAT107 | Activity | 0 | ALA3089296 | Active | Homo sapiens | |||||
5. | ALA3086473 | 1a, GAT106 | Activity | 0 | ALA3089295 | Not Active | Homo sapiens | |||||
6. | ALA3086472 | 1b, GAT107 | EC50 | = | 28 | uM | ALA3089294 | 4.55 | nM | Homo sapiens | ||
7. | ALA3086472 | 1b, GAT107 | Activity | 0 | ALA3089293 | Dose-dependent effect | Homo sapiens | |||||
8. | ALA3086472 | 1b, GAT107 | Activity | 0 | ALA3089292 | Active | Homo sapiens | |||||
9. | ALA3086472 | 1b, GAT107 | Activity | 0 | ALA3089291 | Active | Homo sapiens | |||||
10. | ALA3086474 | 1, Cis diastereomer | Activity | 0 | ALA3089290 | Active | Homo sapiens | |||||
11. | ALA3086472 | 1b, GAT107 | Activity | 0 | ALA3089290 | Active | Homo sapiens | |||||
12. | ALA3086472 | 1b, GAT107 | Activity | 0 | ALA3089287 | Active | Homo sapiens | |||||
13. | ALA965 | SID11110943 | Ki | = | 66 | uM | ALA2445786 | 4.18 | nM | Homo sapiens | ||
14. | ALA1472561 | SID11111411 | Ki | = | 44 | uM | ALA2445786 | 4.36 | nM | Homo sapiens | ||
15. | ALA2441748 | DMCC | Ki | 0 | ALA2445786 | Not Determined | Homo sapiens | |||||
16. | ALA2441749 | 59 | Ki | 0 | ALA2445786 | Not Determined | Homo sapiens | |||||
17. | bethanechol | bethanechol | Ki | 0 | ALA2445786 | Not Determined | Homo sapiens | |||||
18. | ALA2440297 | 7p | EC50 | = | 2.5 | uM | ALA2447428 | 5.60 | nM | Homo sapiens | ||
19. | ALA2440120 | 7b | EC50 | = | 1.9 | uM | ALA2447428 | 5.72 | nM | Homo sapiens | ||
20. | ALA2440296 | 7q | EC50 | = | 0.38 | uM | ALA2447428 | 6.42 | nM | Homo sapiens |