| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  A 485 | A-485 | Cell Proliferation EC50 | 1.063 | uM | ALA4886695 | uM | Homo sapiens | ||||
| 2. |  2-methyl-N-[2-({3-[2-(prop-2-enamido)acetamido]phenyl}amino)pyrimidin-5-yl]-5-[3-(trifluoromethyl)benzamido]benzamide | 38 | RatioGI50 | = | 35 | ALA3292717 | Homo sapiens | |||||
| 3. |  2-methyl-N-(2-{[3-(prop-2-enamido)phenyl]amino}pyrimidin-5-yl)-5-[3-(trifluoromethyl)benzamido]benzamide | 31 | RatioGI50 | = | 35 | ALA3292717 | Homo sapiens | |||||
| 4. |  Ibrutinib (PCI-32765) | SID124898784 | GI50 | = | 1.09 | uM | ALA3292459 | nM | Homo sapiens | |||
| 5. | 2-methyl-N-[2-({3-[2-(prop-2-enamido)acetamido]phenyl}amino)pyrimidin-5-yl]-5-[3-(trifluoromethyl)benzamido]benzamide | 38 | GI50 | = | 0.029 | uM | ALA3292459 | nM | Homo sapiens | |||
| 6. | 2-methyl-N-(2-{[3-(prop-2-enamido)phenyl]amino}pyrimidin-5-yl)-5-[3-(trifluoromethyl)benzamido]benzamide | 31 | GI50 | = | 0.031 | uM | ALA3292459 | nM | Homo sapiens | |||
| 7. |  ALA3331534 | 19 | GI50 | = | 2.7 | uM | ALA3388646 | nM | Homo sapiens | |||
| 8. | ALA3331534 | 19 | GI50 | = | 3.7 | uM | ALA3388050 | nM | Homo sapiens | |||
| 9. |  ALA4462577 | 36 | IC50 | = | 0.005 | uM | ALA5116373 | 8.28 | nM | Homo sapiens | ||
| 10. |  ALA191384 | figure 1, 6 | IC50 | = | 10.244 | uM | ALA2363824 | 4.99 | nM | Homo sapiens | ||
| 11. |  ALA289228 | 1, R-115777 | IC50 | = | 21.166 | uM | ALA2363824 | 4.67 | nM | Homo sapiens | ||
| 12. |  Epothilone B | Epothilone B | IC50 | = | 0.004 | uM | ALA2363824 | 8.38 | nM | Homo sapiens | ||
| 13. |  Pazopanib | 13 | IC50 | = | 352.549 | uM | ALA2363824 | nM | Homo sapiens | |||
| 14. |  Bryostatin 1 | bryostatin 1 | IC50 | = | 0.217 | uM | ALA2363824 | 6.66 | nM | Homo sapiens | ||
| 15. |  ALA252164 | 40f, VER-52296, NVP-AUY922 | IC50 | = | 0.073 | uM | ALA2363824 | 7.13 | nM | Homo sapiens | ||
| 16. |  LFM-A13 | LFM-A13 | IC50 | = | 376.735 | uM | ALA2363824 | nM | Homo sapiens | |||
| 17. |  ALA403664 | blenoxane | IC50 | = | 31.634 | uM | ALA2363824 | 4.50 | nM | Homo sapiens | ||
| 18. |  Bexarotene | LGD-1069 | IC50 | = | 1069.702 | uM | ALA2363824 | nM | Homo sapiens | |||
| 19. |  ALA1091644 | OSI-906 | IC50 | = | 22.158 | uM | ALA2363824 | 4.65 | nM | Homo sapiens | ||
| 20. |  BMS-754807 | 9d, BMS-754807 | IC50 | = | 12.379 | uM | ALA2363824 | 4.91 | nM | Homo sapiens |
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