# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Rotenone | 1 | IC50 | = | 0.3 | uM | ALA2411683 | 6.52 | nM | Homo sapiens | ||
2. | Tephrosin | 13 (tephrosin) | IC50 | = | 5.4 | uM | ALA2411683 | 5.27 | nM | Homo sapiens | ||
3. | ALA240545 | 4, 12a-hydroxyrotenone | IC50 | = | 0.5 | uM | ALA2411681 | 6.30 | nM | Homo sapiens | ||
4. | Rotenone | 1 | IC50 | = | 0.3 | uM | ALA2411681 | 6.52 | nM | Homo sapiens | ||
5. | Tephrosin | 13 (tephrosin) | IC50 | = | 9 | uM | ALA2411681 | 5.05 | nM | Homo sapiens | ||
6. | Tephrosin | 13 (tephrosin) | Activity | = | 24 | % | ALA2411677 | % | Homo sapiens | |||
7. | Tephrosin | 13 (tephrosin) | Activity | 0 | ALA2411676 | Active | Homo sapiens | |||||
8. | ALA240545 | 4, 12a-hydroxyrotenone | IC50 | = | 0.7 | uM | ALA2411683 | 6.16 | nM | Homo sapiens | ||
9. | ALA1614701 | AZD-6244 | IC50 | = | 6.674 | uM | ALA2363713 | 5.18 | nM | Homo sapiens | ||
10. | SB590885 | 33, SB-590885 | IC50 | = | 5.583 | uM | ALA2363713 | 5.25 | nM | Homo sapiens | ||
11. | PD0325901 | 34, PD-0325901 | IC50 | = | 13.007 | uM | ALA2363713 | 4.89 | nM | Homo sapiens | ||
12. | AZD8055 | 10, AZD-8055 | IC50 | = | 0.274 | uM | ALA2363713 | 6.56 | nM | Homo sapiens | ||
13. | GDC-0941 | 17, GDC-0941 | IC50 | = | 0.832 | uM | ALA2363713 | 6.08 | nM | Homo sapiens | ||
14. | BEZ235 | SID124898663 | IC50 | = | 0.017 | uM | ALA2363713 | 7.76 | nM | Homo sapiens | ||
15. | Palbociclib | 43(table 3) | IC50 | = | 0.148 | uM | ALA2363713 | 6.83 | nM | Homo sapiens | ||
16. | MK-2206 | 17 | IC50 | = | 1.376 | uM | ALA2363713 | 5.86 | nM | Homo sapiens | ||
17. | Ro 3306 | 28 | IC50 | = | 170.815 | uM | ALA2363713 | nM | Homo sapiens | |||
18. | ZM-447439 | 2 | IC50 | = | 0.739 | uM | ALA2363713 | 6.13 | nM | Homo sapiens | ||
19. | PD173074 | 12 | IC50 | = | 2.653 | uM | ALA2363713 | 5.58 | nM | Homo sapiens | ||
20. | Nutlin-3a | Nutlin-3 | IC50 | = | 5.446 | uM | ALA2363713 | 5.26 | nM | Homo sapiens |