# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5218950 | 29f; VU6027634 | IC50 | > | 10000 | nM | ALA5216724 | nM | Rattus norvegicus | |||
2. | ALA5218449 | (rac)-30c; VU6035461 | IC50 | = | 300 | nM | ALA5216724 | 6.52 | nM | Rattus norvegicus | ||
3. | ALA5218711 | (rac)-30b; VU6035460 | IC50 | = | 110 | nM | ALA5216724 | 6.96 | nM | Rattus norvegicus | ||
4. | ALA5218950 | 29f; VU6027634 | Activity | = | 35 | % | ALA5216716 | % | Rattus norvegicus | |||
5. | ALA5218449 | (rac)-30c; VU6035461 | Activity | = | 3 | % | ALA5216716 | % | Rattus norvegicus | |||
6. | ALA5218711 | (rac)-30b; VU6035460 | Activity | = | 3 | % | ALA5216716 | % | Rattus norvegicus | |||
7. | ALA5204021 | 27b; VU6019650 | IC50 | = | 2.2 | nM | ALA5164551 | 8.66 | nM | Rattus norvegicus | ||
8. | ALA5189893 | 19; VU6015241 | IC50 | > | 10000 | nM | ALA5133244 | nM | Rattus norvegicus | |||
9. | PF-06767832 | 7; PF-06767832 | Activity | 0 | ALA4717813 | Dose-dependent effect | Rattus norvegicus | |||||
10. | PF-06767832 | 7; PF-06767832 | Activity | 0 | ALA4717812 | Dose-dependent effect | Rattus norvegicus | |||||
11. | ALA4248057 | VU6007318; 14a | %max | = | 87 | % | ALA4237183 | % | Rattus norvegicus | |||
12. | ALA4248057 | VU6007318; 14a | EC50 | = | 0.04 | uM | ALA4237183 | 7.40 | nM | Rattus norvegicus | ||
13. | ALA4248057 | VU6007318; 14a | pEC50 | = | 7.41 | ALA4237183 | 7.41 | nM | Rattus norvegicus | |||
14. | ALA4247625 | 14b | %max | = | 86 | % | ALA4237183 | % | Rattus norvegicus | |||
15. | ALA4247625 | 14b | EC50 | = | 0.014 | uM | ALA4237183 | 7.85 | nM | Rattus norvegicus | ||
16. | ALA4247625 | 14b | pEC50 | = | 7.86 | ALA4237183 | 7.86 | nM | Rattus norvegicus | |||
17. | ALA4237601 | VU6007661; 14c | %max | = | 90 | % | ALA4237183 | % | Rattus norvegicus | |||
18. | ALA4237601 | VU6007661; 14c | EC50 | = | 0.1 | uM | ALA4237183 | 7.00 | nM | Rattus norvegicus | ||
19. | ALA4237601 | VU6007661; 14c | pEC50 | = | 7 | ALA4237183 | 7.00 | nM | Rattus norvegicus | |||
20. | ALA4246159 | 15a | %max | = | 87 | % | ALA4237183 | % | Rattus norvegicus |