# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4847762 | 14f | TGI | = | 48.7 | % | ALA4841363 | % | Homo sapiens | |||
2. | BI-D1870 | BI-D1870 | TGI | = | 41.6 | % | ALA4841363 | % | Homo sapiens | |||
3. | ALA4847762 | 14f | TGI | = | 73.4 | % | ALA4841362 | % | Homo sapiens | |||
4. | ALA4847762 | 14f | Ratio IC50 | = | 8 | ALA4841361 | Homo sapiens | |||||
5. | ALA4847762 | 14f | INH | 0 | ALA4841360 | Dose-Dependent Effect | % | Homo sapiens | ||||
6. | ALA4847762 | 14f | IC50 | = | 0.57 | uM | ALA4841360 | 6.24 | nM | Homo sapiens | ||
7. | BI-D1870 | BI-D1870 | IC50 | = | 4.553 | uM | ALA4841360 | 5.34 | nM | Homo sapiens | ||
8. | ALA4847762 | 14f | Ratio IC50 | = | 2 | ALA4841359 | Homo sapiens | |||||
9. | ALA4847762 | 14f | IC50 | = | 0.983 | uM | ALA4841358 | 6.01 | nM | Homo sapiens | ||
10. | BI-D1870 | BI-D1870 | IC50 | = | 1.89 | uM | ALA4841358 | 5.72 | nM | Homo sapiens | ||
11. | Rucaparib | 63, AG-014699 | IC50 | = | 29.812 | uM | ALA2363788 | 4.53 | nM | Homo sapiens | ||
12. | CCT 018159 | 3a CCT018159 | IC50 | = | 27.021 | uM | ALA2363788 | 4.57 | nM | Homo sapiens | ||
13. | TW-37 | 5, TW-37 | IC50 | = | 1.234 | uM | ALA2363788 | 5.91 | nM | Homo sapiens | ||
14. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 21.063 | uM | ALA2363788 | 4.68 | nM | Homo sapiens | ||
15. | PF-4708671 | SID137275978 | IC50 | = | 170.252 | uM | ALA2363788 | nM | Homo sapiens | |||
16. | Avagacestat | 80 BMS-708163 | IC50 | = | 492.819 | uM | ALA2363788 | nM | Homo sapiens | |||
17. | EHT 1864 | SID137275837 | IC50 | = | 953.321 | uM | ALA2363788 | nM | Homo sapiens | |||
18. | CCT007093 | A17 | IC50 | = | 570.145 | uM | ALA2363788 | nM | Homo sapiens | |||
19. | AZD6482 | AZD-6482 | IC50 | = | 19.659 | uM | ALA2363788 | 4.71 | nM | Homo sapiens | ||
20. | ALA1614701 | AZD-6244 | IC50 | = | 27.636 | uM | ALA2363788 | 4.56 | nM | Homo sapiens |