# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Pyridone 6 | 6 | IC50 | = | 250 | nM | ALA5245518 | 6.60 | nM | Homo sapiens | ||
2. | ALA3973951 | 8f | IC50 | = | 40.61 | uM | ALA5241880 | 4.39 | nM | Homo sapiens | ||
3. | Ebselen | Ebselen | IC50 | = | 40 | uM | ALA5237174 | 4.40 | nM | Homo sapiens | ||
4. | ALA301982 | 1 | IC50 | = | 0.47 | uM | ALA5233848 | 6.33 | nM | Homo sapiens | ||
5. | ALA5287361 | 15b | IC50 | = | 1.2 | uM | ALA5230963 | 5.92 | nM | Homo sapiens | ||
6. | ALA5281688 | 15a | IC50 | = | 1.2 | uM | ALA5230963 | 5.92 | nM | Homo sapiens | ||
7. | ALA4215914 | 9 | IC50 | = | 5 | uM | ALA5230785 | 5.30 | nM | Homo sapiens | ||
8. | Rocilinostat (ACY-1215) | RICOLINOSTAT | IC50 | > | 100 | uM | ALA5230353 | nM | Homo sapiens | |||
9. | Vorinostat (SAHA, MK0683) | SAHA | IC50 | = | 0.59 | uM | ALA5230353 | 6.23 | nM | Homo sapiens | ||
10. | ALA5268638 | 21b | IC50 | = | 43.233 | uM | ALA5230353 | 4.36 | nM | Homo sapiens | ||
11. | ALA5266137 | 18d | IC50 | = | 23.1 | uM | ALA5230353 | 4.64 | nM | Homo sapiens | ||
12. | ALA5286689 | 18b | IC50 | = | 23.37 | uM | ALA5230353 | 4.63 | nM | Homo sapiens | ||
13. | ALA5289315 | 18a | IC50 | = | 25.882 | uM | ALA5230353 | 4.59 | nM | Homo sapiens | ||
14. | ALA5273674 | 11b | IC50 | = | 86.34 | uM | ALA5230353 | 4.06 | nM | Homo sapiens | ||
15. | SKLB-23bb | 23bb | IC50 | = | 31 | nM | ALA5227765 | 7.51 | nM | Homo sapiens | ||
16. | ALA5190272 | AG6033 | Activity | 0 | ALA5164472 | NA | Homo sapiens | |||||
17. | ALA5196874 | (-)-53; MU1656 | Activity | 0 | ALA5162058 | NA | Homo sapiens | |||||
18. | M3258 | 50 | Activity | 0 | ALA5151730 | NA | Homo sapiens | |||||
19. | M3258 | 50 | Activity | 0 | ALA5151729 | Active | Homo sapiens | |||||
20. | M3258 | 50 | Activity | 0 | ALA5151728 | Active | Homo sapiens |