# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3348846 | SID174006594 | IC50 | = | 83.6 | nM | ALA5251053 | 7.08 | nM | Homo sapiens | ||
2. | ALA5274338 | 2e | IC50 | = | 299.5 | nM | ALA5251053 | 6.52 | nM | Homo sapiens | ||
3. | Tapotoclax | 2; AMG 176 | INH | = | 99 | % | ALA5242718 | % | Homo sapiens | |||
4. | ALA5196874 | (-)-53; MU1656 | Activity | 0 | ALA5162027 | NA | Homo sapiens | |||||
5. | ALA5177205 | 1u | Activity | = | 38.27 | % | ALA5124286 | % | Homo sapiens | |||
6. | ALA5186832 | 1l | Activity | = | 28.49 | % | ALA5124286 | % | Homo sapiens | |||
7. | SGC-CBP30 | 72 | Activity | 0 | ALA5124286 | NA | Homo sapiens | |||||
8. | ALA5177205 | 1u | Activity | = | 90 | % | ALA5124285 | % | Homo sapiens | |||
9. | ALA5186832 | 1l | Activity | = | 90 | % | ALA5124285 | % | Homo sapiens | |||
10. | SGC-CBP30 | 72 | Activity | 0 | ALA5124285 | NA | Homo sapiens | |||||
11. | ALA5189469 | 1v | IC50 | = | 1.54 | uM | ALA5124276 | 5.81 | nM | Homo sapiens | ||
12. | ALA5177205 | 1u | IC50 | = | 1.09 | uM | ALA5124276 | 5.96 | nM | Homo sapiens | ||
13. | ALA5186832 | 1l | IC50 | = | 1.39 | uM | ALA5124276 | 5.86 | nM | Homo sapiens | ||
14. | ALA5193321 | 1k | IC50 | = | 2.29 | uM | ALA5124276 | 5.64 | nM | Homo sapiens | ||
15. | SGC-CBP30 | 72 | IC50 | = | 2.64 | uM | ALA5124276 | 5.58 | nM | Homo sapiens | ||
16. | ALA1898589 | SID99355980 | IC50 | = | 4 | uM | ALA4418233 | 5.40 | nM | Homo sapiens | ||
17. | ALA4077014 | 3g | IC50 | = | 0.3 | uM | ALA4418233 | 6.52 | nM | Homo sapiens | ||
18. | ALA1898589 | SID99355980 | Activity | 0 | ALA4418234 | Active | Homo sapiens | |||||
19. | ALA4077014 | 3g | Activity | 0 | ALA4418234 | Active | Homo sapiens | |||||
20. | ALA4522028 | dMCL1-2 | Activity | 0 | ALA4398186 | Toxic | Homo sapiens |