# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5196874 | (-)-53; MU1656 | Activity | 0 | ALA5161989 | NA | Homo sapiens | |||||
2. | 2-methyl-N-(2-{[3-(prop-2-enamido)phenyl]amino}pyrimidin-5-yl)-5-[3-(trifluoromethyl)benzamido]benzamide | 31 | GI | 0 | ALA3292451 | Active | Homo sapiens | |||||
3. | ALA1614701 | AZD-6244 | IC50 | = | 0.701 | uM | ALA2363322 | 6.16 | nM | Homo sapiens | ||
4. | SB590885 | 33, SB-590885 | IC50 | = | 12.093 | uM | ALA2363322 | 4.92 | nM | Homo sapiens | ||
5. | PD0325901 | 34, PD-0325901 | IC50 | = | 0.286 | uM | ALA2363322 | 6.54 | nM | Homo sapiens | ||
6. | AZD8055 | 10, AZD-8055 | IC50 | = | 0.463 | uM | ALA2363322 | 6.33 | nM | Homo sapiens | ||
7. | GDC-0941 | 17, GDC-0941 | IC50 | = | 1.649 | uM | ALA2363322 | 5.78 | nM | Homo sapiens | ||
8. | BEZ235 | SID124898663 | IC50 | = | 0.031 | uM | ALA2363322 | 7.51 | nM | Homo sapiens | ||
9. | Palbociclib | 43(table 3) | IC50 | = | 0.852 | uM | ALA2363322 | 6.07 | nM | Homo sapiens | ||
10. | MK-2206 | 17 | IC50 | = | 8.153 | uM | ALA2363322 | 5.09 | nM | Homo sapiens | ||
11. | Ro 3306 | 28 | IC50 | = | 14.263 | uM | ALA2363322 | 4.85 | nM | Homo sapiens | ||
12. | ZM-447439 | 2 | IC50 | = | 2.748 | uM | ALA2363322 | 5.56 | nM | Homo sapiens | ||
13. | PD173074 | 12 | IC50 | = | 44.053 | uM | ALA2363322 | 4.36 | nM | Homo sapiens | ||
14. | Nutlin-3a | Nutlin-3 | IC50 | = | 2.593 | uM | ALA2363322 | 5.59 | nM | Homo sapiens | ||
15. | Wee1 inhibitor | 23 | IC50 | = | 1.431 | uM | ALA2363322 | 5.84 | nM | Homo sapiens | ||
16. | TCS JNK 6o | 6o | IC50 | = | 252.057 | uM | ALA2363322 | nM | Homo sapiens | |||
17. | Doramapimod | 45 | IC50 | = | 57.451 | uM | ALA2363322 | 4.24 | nM | Homo sapiens | ||
18. | BI-D1870 | BI-D1870 | IC50 | = | 3.068 | uM | ALA2363322 | 5.51 | nM | Homo sapiens | ||
19. | SL 0101-1 | 1, SL-0101 | IC50 | = | 250.702 | uM | ALA2363322 | nM | Homo sapiens | |||
20. | NU7441 (KU-57788) | 22g | IC50 | = | 3.481 | uM | ALA2363322 | 5.46 | nM | Homo sapiens |