# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Azelastine | Azelastine | IC50 | = | 8 | uM | ALA3638170 | 5.10 | Original reference for datapoint is pubmed_id: 7957608 | nM | Cavia porcellus | |
2. | Ropivacaine base | Ropivacaine | IC50 | = | 430 | uM | ALA3638169 | Original reference for datapoint is pubmed_id: 14517618 | nM | Cavia porcellus | ||
3. | Arecoline | arecoline | IC50 | = | 33.73 | uM | ALA3638167 | 4.47 | Original reference for datapoint is pubmed_id: 12674757 | nM | Cavia porcellus | |
4. | ALA408 | Troglitazone | IC50 | = | 0.8 | uM | ALA3638163 | 6.10 | Original reference for datapoint is pubmed_id: 10877527 | nM | Cavia porcellus | |
5. | ALA363295 | Terodiline | IC50 | = | 33.5 | uM | ALA3638159 | 4.47 | Original reference for datapoint is pubmed_id: 9151306 | nM | Cavia porcellus | |
6. | ALA3638053 | RCC-36 | IC50 | = | 27 | uM | ALA3638158 | 4.57 | Original reference for datapoint is pubmed_id: 9151306 | nM | Cavia porcellus | |
7. | ALA2107463 | TEMIVERINE | IC50 | = | 27 | uM | ALA3638157 | 4.57 | Original reference for datapoint is pubmed_id: 9151306 | nM | Cavia porcellus | |
8. | bepridil | Bepridil | IC50 | = | 1.55 | uM | ALA3638155 | 5.81 | Original reference for datapoint is pubmed_id: 8591000 | nM | Cavia porcellus | |
9. | ALA2105033 | LEVOSEMOTIADIL | IC50 | = | 1.29 | uM | ALA3638154 | 5.89 | Original reference for datapoint is pubmed_id: 8591000 | nM | Cavia porcellus | |
10. | thiopental | thiopental | IC50 | = | 0.28 | uM | ALA3638153 | 6.55 | Original reference for datapoint is pubmed_id: 17519531 | nM | Cavia porcellus | |
11. | mepacrine | quinacrine | IC50 | = | 5.6 | uM | ALA3638152 | 5.25 | Original reference for datapoint is pubmed_id: 8791171 | nM | Cavia porcellus | |
12. | Celecoxib | Celecoxib | IC50 | = | 10.6 | uM | ALA3638151 | 4.97 | Original reference for datapoint is pubmed_id: 25889233 | nM | Cavia porcellus | |
13. | ALA3638051 | Sulcardine | IC50 | = | 69.2 | uM | ALA3638138 | 4.16 | Original reference for datapoint is pubmed_id: 22922342 | nM | Cavia porcellus | |
14. | ALA1078261 | Propiverine | IC50 | = | 34.7 | uM | ALA3638133 | 4.46 | Original reference for datapoint is pubmed_id: 18092154 | nM | Cavia porcellus | |
15. | Verapamil | 24 | IC50 | = | 1.5 | uM | ALA3638130 | 5.82 | Original reference for datapoint is pubmed_id: 23396228 | nM | Cavia porcellus | |
16. | Caffeic acid phenethyl ester | CAPE | IC50 | = | 1.1 | uM | ALA3638129 | 5.96 | Original reference for datapoint is pubmed_id: 23396228 | nM | Cavia porcellus | |
17. | dronedarone | Dronedarone | IC50 | = | 0.4 | uM | ALA3638128 | 6.40 | Original reference for datapoint is pubmed_id: 21279331 | nM | Cavia porcellus | |
18. | ALA3638037 | Cinnamophilin | IC50 | = | 7.5 | uM | ALA3638097 | 5.12 | max inhibition = 104%. Original reference for datapoint is pubmed_id: 17965733 | nM | Cavia porcellus | |
19. | Sipatrigine | 30 | IC50 | = | 6.02 | uM | ALA3638096 | 5.22 | Original reference for datapoint is pubmed_id: 16445575 | nM | Cavia porcellus | |
20. | cyproheptadine | 7 | IC50 | = | 7.75 | uM | ALA3638091 | 5.11 | Original reference for datapoint is pubmed_id: 12686765 | nM | Cavia porcellus |