# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4462318 | 19i | Kd(free) | = | 2.296 | uM | ALA4371428 | 5.64 | nM | Homo sapiens | ||
2. | ALA4443828 | 19h | Kd(free) | = | 1.078 | uM | ALA4371428 | 5.97 | nM | Homo sapiens | ||
3. | Imatinib (STI571) | 1 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
4. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
5. | Abemaciclib | ABEMACICLIB | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
6. | AZD6482 | AZD-6482 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
7. | GSK1070916 | GSK-1070916 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
8. | ALA3544944 | XL-413 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
9. | PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
10. | JANEX-1 | JANEX-1 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
11. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
12. | LY2603618 | RABUSERTIB | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
13. | MK-8776 (SCH 900776) | 29 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
14. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
15. | AZD1208 | 28 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
16. | ASP3026 | ASP-3026 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
17. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
18. | LY2157299 | GALUNISERTIB | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
19. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens | ||
20. | LY2584702 | LY-2584702 | Kd apparent | > | 30000 | nM | ALA3991840 | Inactive | nM | Homo sapiens |