# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2288594 | 2d-trans enantiomer I | INH | 0 | ALA3073734 | Active | % | Bos taurus | ||||
2. | ALA417295 | 2e, racemic mixture of trans and cis diastereomers | INH | 0 | ALA3073734 | Active | % | Bos taurus | ||||
3. | Colchicine | colchicine | INH | 0 | ALA3073733 | Active | % | Bos taurus | ||||
4. | Colchicine | colchicine | EC50 | = | 0.75 | uM | ALA3073731 | 6.12 | nM | Bos taurus | ||
5. | ALA32082 | 2b, racmixture of trans diastereomer | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
6. | ALA282958 | 2c, racemic mixture of trans diastereomer | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
7. | ALA2288594 | 2d-trans enantiomer I | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
8. | ALA417295 | 2e, racemic mixture of trans and cis diastereomers | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
9. | ALA2288594 | 2d-trans enantiomer I | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
10. | ALA2288594 | 2d-trans enantiomer I | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
11. | ALA2288593 | 2e-cis enantiomer II | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
12. | ALA2288593 | 2e-cis enantiomer II | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
13. | ALA2288592 | 2e-trans enantiomer II | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
14. | ALA2288592 | 2e-trans enantiomer II | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
15. | ALA32021 | 3a | EC50 | > | 100 | uM | ALA3073731 | nM | Bos taurus | |||
16. | ALA32128 | 3b | EC50 | = | 50 | uM | ALA3073731 | 4.30 | nM | Bos taurus | ||
17. | ALA31779 | 3c | EC50 | = | 6.25 | uM | ALA3073731 | 5.20 | nM | Bos taurus | ||
18. | ALA31663 | 3d | EC50 | = | 6.25 | uM | ALA3073731 | 5.20 | nM | Bos taurus | ||
19. | ALA32242 | 3e | EC50 | = | 6.25 | uM | ALA3073731 | 5.20 | nM | Bos taurus | ||
20. | ALA28250 | SID87335404 | EC50 | = | 6.25 | uM | ALA3073731 | 5.20 | nM | Bos taurus |